Tekturna
Hypertensive disease, not adequately controlled with monotherapy
Treatment
2 FDA approvals
20 Active Studies for Tekturna
Treatment for
Hypertensive disease
What is Tekturna
Aliskiren
The Generic name of this drug
Treatment Summary
Aliskiren is a medication used to treat high blood pressure. It was developed by Speedel and Novartis and approved by the FDA in 2007. Aliskiren works by blocking an enzyme known as renin and can be used on its own or in combination with other medications to reduce blood pressure.
Tekturna
is the brand name
Tekturna Overview & Background
Brand Name
Generic Name
First FDA Approval
How many FDA approvals?
Tekturna
Aliskiren
2007
36
Approved as Treatment by the FDA
Aliskiren, also known as Tekturna, is approved by the FDA for 2 uses including Hypertensive disease and not adequately controlled with monotherapy .
Hypertensive disease
Used to treat High Blood Pressure (Hypertension) in combination with Amlodipine
not adequately controlled with monotherapy
Used to treat not adequately controlled with monotherapy in combination with Hydrochlorothiazide
Effectiveness
How Tekturna Affects Patients
Aliskiren lowers blood pressure by blocking the enzyme renin. This has a chain reaction that results in lower blood pressure, which can help prevent life-threatening and non-deadly cardiovascular issues such as stroke and heart attack.
How Tekturna works in the body
Aliskiren is a drug that helps lower blood pressure by blocking the action of a protein called renin. Normally, when blood volume and renal perfusion decrease, renin is released from the kidneys. Renin then turns a protein called angiotensinogen into angiotensin I, which is then converted to angiotensin II. Angiotensin II is a hormone that causes blood vessels to constrict, which increases blood pressure. Aliskiren works by binding to renin and preventing it from turning angiotensinogen into angiotensin I, thereby stopping the release of angiotensin II
When to interrupt dosage
The amount of Tekturna is subject to the diagnosed state. The dosage amount shifts as per the system of delivery (e.g. Oral or Tablet, film coated) provided in the table beneath.
Condition
Dosage
Administration
not adequately controlled with monotherapy
300.0 mg, 150.0 mg,
Tablet, film coated - Oral, , Oral, Tablet, film coated, Tablet - Oral, Tablet
Hypertensive disease
300.0 mg, 150.0 mg,
Tablet, film coated - Oral, , Oral, Tablet, film coated, Tablet - Oral, Tablet
Warnings
Tekturna has four counterindications and should not be ingested when confronting any of the conditions given in the following table.
Tekturna Contraindications
Condition
Risk Level
Notes
Pulse Frequency
Do Not Combine
Pulse Frequency
Do Not Combine
Type 2 Diabetes
Do Not Combine
Type 2 Diabetes
Do Not Combine
There are 20 known major drug interactions with Tekturna.
Common Tekturna Drug Interactions
Drug Name
Risk Level
Description
Amifostine
Major
Aliskiren may increase the hypotensive activities of Amifostine.
Azilsartan medoxomil
Major
Aliskiren may increase the hypotensive and hyperkalemic activities of Azilsartan medoxomil.
Benazepril
Major
The risk or severity of hypotension, hyperkalemia, and nephrotoxicity can be increased when Aliskiren is combined with Benazepril.
Benazeprilat
Major
The risk or severity of hypotension, hyperkalemia, and nephrotoxicity can be increased when Aliskiren is combined with Benazeprilat.
Captopril
Major
The risk or severity of hypotension, hyperkalemia, and nephrotoxicity can be increased when Aliskiren is combined with Captopril.
Tekturna Toxicity & Overdose Risk
The lowest toxic dose of aliskiren in rats has been found to be greater than 2000mg/kg. If someone takes too much aliskiren, they may experience low blood pressure, and should receive supportive treatment.
Tekturna Novel Uses: Which Conditions Have a Clinical Trial Featuring Tekturna?
18 active studies are currently investigating the potential of Tekturna in ameliorating Hypertensive diseases.
Condition
Clinical Trials
Trial Phases
Hypertensive disease
27 Actively Recruiting
Not Applicable, Phase 1, Phase 2, Phase 3
not adequately controlled with monotherapy
0 Actively Recruiting
Tekturna Reviews: What are patients saying about Tekturna?
5
Patient Review
8/13/2015
Tekturna for High Blood Pressure
5
Patient Review
8/30/2012
Tekturna for High Blood Pressure
5
Patient Review
9/25/2011
Tekturna for High Blood Pressure
5
Patient Review
6/5/2013
Tekturna for High Blood Pressure
4.3
Patient Review
4/14/2015
Tekturna for High Blood Pressure
4
Patient Review
12/7/2011
Tekturna for High Blood Pressure
3.7
Patient Review
2/12/2012
Tekturna for High Blood Pressure
3.7
Patient Review
12/14/2011
Tekturna for High Blood Pressure
3.3
Patient Review
3/15/2012
Tekturna for High Blood Pressure
3
Patient Review
1/28/2012
Tekturna for High Blood Pressure
2.7
Patient Review
1/19/2012
Tekturna for High Blood Pressure
2.7
Patient Review
7/9/2012
Tekturna for High Blood Pressure
2.3
Patient Review
12/27/2011
Tekturna for High Blood Pressure
2.3
Patient Review
9/25/2011
Tekturna for High Blood Pressure
2.3
Patient Review
12/17/2011
Tekturna for High Blood Pressure
1.3
Patient Review
1/13/2012
Tekturna for High Blood Pressure
Patient Q&A Section about tekturna
These questions and answers are submitted by anonymous patients, and have not been verified by our internal team.
Is Tekturna still on the market?
"The FDA does not recommend that people with diabetes who are taking angiotensin converting enzyme (ACE) inhibitors and angiotensin receptor blockers (ARBs) take Tekturna."
Answered by AI
What is Tekturna prescribed for?
"It is manufactured by the Swiss pharmaceutical company, Novartis.
Tekturna is a medication that lowers blood pressure, used to treat hypertension. It is manufactured by the Swiss pharmaceutical company, Novartis."
Answered by AI
Is Tekturna and ACE inhibitor?
"A product called aliskiren (Tekturna, Rasilez, Novartis) does not have the same effect as an ACE-inhibitor. An ACE-inhibitor prevents the breakdown of bradykinin. Increased levels of bradykinin cause the release of local vasodilators and may be part of the additional protective benefit of ACE-inhibitors."
Answered by AI
What type of drug is Tekturna?
"Tekturna is the first FDA-approved drug in a new class of high blood pressure drugs that work by inhibiting the production of renin, an enzyme produced by the kidneys. Renin helps to regulate blood pressure and its overproduction can lead to higher blood pressure."
Answered by AI