Arestin
Rocky Mountain Spotted Fever, Relapsing Fever, Trachoma + 22 more
Treatment
5 Active Studies for Arestin
Treatment for
Rocky Mountain Spotted Fever
What is Arestin
Minocycline
The Generic name of this drug
Treatment Summary
Minocycline is an antibiotic that was developed in 1966. It is more powerful than other tetracycline antibiotics and works to kill both gram-positive and gram-negative bacteria. It was approved by the FDA in 1971 and is commonly used to treat infections.
Minocin
is the brand name
Arestin Overview & Background
Brand Name
Generic Name
First FDA Approval
How many FDA approvals?
Minocin
Minocycline
1990
305
Effectiveness
How Arestin Affects Patients
Minocycline is an antibiotic that stops bacteria from making proteins needed for them to survive. It is usually taken 2-4 times a day, so it does not last very long. It should not be taken more than 400mg in 24 hours. People should be aware of the potential risks associated with taking minocycline, such as problems with teeth and bone development, inflammation of the colon, side effects on the central nervous system, and swelling of the brain.
How Arestin works in the body
Tetracyclines enter bacteria by attaching to metal ions like magnesium. This allows the medicine to enter the bacteria's outer membrane and dissolve, allowing it to pass into the cytoplasm. Once inside, tetracyclines prevent proteins from being formed, stopping the bacteria from reproducing.
When to interrupt dosage
The quantity of Arestin is contingent upon the diagnosed condition, including Periodontitis, Rickettsialpox and Lymphogranuloma Venereum. The amount of dosage is contingent upon the technique of delivery (e.g. Capsule, extended release or Tablet, film coated, extended release) noted in the following table.
Condition
Dosage
Administration
Brucellosis
, 75.0 mg, 45.0 mg, 90.0 mg, 135.0 mg, 50.0 mg, 100.0 mg, 80.0 mg, 1.0 mg, 65.0 mg, 115.0 mg, 55.0 mg, 105.0 mg, 67.5 mg, 112.5 mg, 0.04 mg/mg, 0.015 mg/mg, 1.0 mg/mg
, Oral, Capsule - Oral, Capsule, Tablet, extended release, Tablet, extended release - Oral, Capsule, extended release, Capsule, extended release - Oral, Kit, Tablet - Oral, Tablet, Tablet, film coated, extended release, Tablet, film coated, extended release - Oral, Intravenous, Injection, Injection - Intravenous, Tablet, film coated, Tablet, film coated - Oral, Powder, Powder - Oral, Capsule, coated pellets, Capsule, coated pellets - Oral, Topical, Aerosol, foam - Topical, Aerosol, foam
Gum Disease
, 75.0 mg, 45.0 mg, 90.0 mg, 135.0 mg, 50.0 mg, 100.0 mg, 80.0 mg, 1.0 mg, 65.0 mg, 115.0 mg, 55.0 mg, 105.0 mg, 67.5 mg, 112.5 mg, 0.04 mg/mg, 0.015 mg/mg, 1.0 mg/mg
, Oral, Capsule - Oral, Capsule, Tablet, extended release, Tablet, extended release - Oral, Capsule, extended release, Capsule, extended release - Oral, Kit, Tablet - Oral, Tablet, Tablet, film coated, extended release, Tablet, film coated, extended release - Oral, Intravenous, Injection, Injection - Intravenous, Tablet, film coated, Tablet, film coated - Oral, Powder, Powder - Oral, Capsule, coated pellets, Capsule, coated pellets - Oral, Topical, Aerosol, foam - Topical, Aerosol, foam
Campylobacter fetus
, 75.0 mg, 45.0 mg, 90.0 mg, 135.0 mg, 50.0 mg, 100.0 mg, 80.0 mg, 1.0 mg, 65.0 mg, 115.0 mg, 55.0 mg, 105.0 mg, 67.5 mg, 112.5 mg, 0.04 mg/mg, 0.015 mg/mg, 1.0 mg/mg
, Oral, Capsule - Oral, Capsule, Tablet, extended release, Tablet, extended release - Oral, Capsule, extended release, Capsule, extended release - Oral, Kit, Tablet - Oral, Tablet, Tablet, film coated, extended release, Tablet, film coated, extended release - Oral, Intravenous, Injection, Injection - Intravenous, Tablet, film coated, Tablet, film coated - Oral, Powder, Powder - Oral, Capsule, coated pellets, Capsule, coated pellets - Oral, Topical, Aerosol, foam - Topical, Aerosol, foam
Psittacosis
, 75.0 mg, 45.0 mg, 90.0 mg, 135.0 mg, 50.0 mg, 100.0 mg, 80.0 mg, 1.0 mg, 65.0 mg, 115.0 mg, 55.0 mg, 105.0 mg, 67.5 mg, 112.5 mg, 0.04 mg/mg, 0.015 mg/mg, 1.0 mg/mg
, Oral, Capsule - Oral, Capsule, Tablet, extended release, Tablet, extended release - Oral, Capsule, extended release, Capsule, extended release - Oral, Kit, Tablet - Oral, Tablet, Tablet, film coated, extended release, Tablet, film coated, extended release - Oral, Intravenous, Injection, Injection - Intravenous, Tablet, film coated, Tablet, film coated - Oral, Powder, Powder - Oral, Capsule, coated pellets, Capsule, coated pellets - Oral, Topical, Aerosol, foam - Topical, Aerosol, foam
Lymphogranuloma Venereum
, 75.0 mg, 45.0 mg, 90.0 mg, 135.0 mg, 50.0 mg, 100.0 mg, 80.0 mg, 1.0 mg, 65.0 mg, 115.0 mg, 55.0 mg, 105.0 mg, 67.5 mg, 112.5 mg, 0.04 mg/mg, 0.015 mg/mg, 1.0 mg/mg
, Oral, Capsule - Oral, Capsule, Tablet, extended release, Tablet, extended release - Oral, Capsule, extended release, Capsule, extended release - Oral, Kit, Tablet - Oral, Tablet, Tablet, film coated, extended release, Tablet, film coated, extended release - Oral, Intravenous, Injection, Injection - Intravenous, Tablet, film coated, Tablet, film coated - Oral, Powder, Powder - Oral, Capsule, coated pellets, Capsule, coated pellets - Oral, Topical, Aerosol, foam - Topical, Aerosol, foam
Granuloma Inguinale
, 75.0 mg, 45.0 mg, 90.0 mg, 135.0 mg, 50.0 mg, 100.0 mg, 80.0 mg, 1.0 mg, 65.0 mg, 115.0 mg, 55.0 mg, 105.0 mg, 67.5 mg, 112.5 mg, 0.04 mg/mg, 0.015 mg/mg, 1.0 mg/mg
, Oral, Capsule - Oral, Capsule, Tablet, extended release, Tablet, extended release - Oral, Capsule, extended release, Capsule, extended release - Oral, Kit, Tablet - Oral, Tablet, Tablet, film coated, extended release, Tablet, film coated, extended release - Oral, Intravenous, Injection, Injection - Intravenous, Tablet, film coated, Tablet, film coated - Oral, Powder, Powder - Oral, Capsule, coated pellets, Capsule, coated pellets - Oral, Topical, Aerosol, foam - Topical, Aerosol, foam
Respiratory Tract Infections
, 75.0 mg, 45.0 mg, 90.0 mg, 135.0 mg, 50.0 mg, 100.0 mg, 80.0 mg, 1.0 mg, 65.0 mg, 115.0 mg, 55.0 mg, 105.0 mg, 67.5 mg, 112.5 mg, 0.04 mg/mg, 0.015 mg/mg, 1.0 mg/mg
, Oral, Capsule - Oral, Capsule, Tablet, extended release, Tablet, extended release - Oral, Capsule, extended release, Capsule, extended release - Oral, Kit, Tablet - Oral, Tablet, Tablet, film coated, extended release, Tablet, film coated, extended release - Oral, Intravenous, Injection, Injection - Intravenous, Tablet, film coated, Tablet, film coated - Oral, Powder, Powder - Oral, Capsule, coated pellets, Capsule, coated pellets - Oral, Topical, Aerosol, foam - Topical, Aerosol, foam
Inflammation
, 75.0 mg, 45.0 mg, 90.0 mg, 135.0 mg, 50.0 mg, 100.0 mg, 80.0 mg, 1.0 mg, 65.0 mg, 115.0 mg, 55.0 mg, 105.0 mg, 67.5 mg, 112.5 mg, 0.04 mg/mg, 0.015 mg/mg, 1.0 mg/mg
, Oral, Capsule - Oral, Capsule, Tablet, extended release, Tablet, extended release - Oral, Capsule, extended release, Capsule, extended release - Oral, Kit, Tablet - Oral, Tablet, Tablet, film coated, extended release, Tablet, film coated, extended release - Oral, Intravenous, Injection, Injection - Intravenous, Tablet, film coated, Tablet, film coated - Oral, Powder, Powder - Oral, Capsule, coated pellets, Capsule, coated pellets - Oral, Topical, Aerosol, foam - Topical, Aerosol, foam
Urethritis
, 75.0 mg, 45.0 mg, 90.0 mg, 135.0 mg, 50.0 mg, 100.0 mg, 80.0 mg, 1.0 mg, 65.0 mg, 115.0 mg, 55.0 mg, 105.0 mg, 67.5 mg, 112.5 mg, 0.04 mg/mg, 0.015 mg/mg, 1.0 mg/mg
, Oral, Capsule - Oral, Capsule, Tablet, extended release, Tablet, extended release - Oral, Capsule, extended release, Capsule, extended release - Oral, Kit, Tablet - Oral, Tablet, Tablet, film coated, extended release, Tablet, film coated, extended release - Oral, Intravenous, Injection, Injection - Intravenous, Tablet, film coated, Tablet, film coated - Oral, Powder, Powder - Oral, Capsule, coated pellets, Capsule, coated pellets - Oral, Topical, Aerosol, foam - Topical, Aerosol, foam
Typhus, Endemic Flea-Borne
, 75.0 mg, 45.0 mg, 90.0 mg, 135.0 mg, 50.0 mg, 100.0 mg, 80.0 mg, 1.0 mg, 65.0 mg, 115.0 mg, 55.0 mg, 105.0 mg, 67.5 mg, 112.5 mg, 0.04 mg/mg, 0.015 mg/mg, 1.0 mg/mg
, Oral, Capsule - Oral, Capsule, Tablet, extended release, Tablet, extended release - Oral, Capsule, extended release, Capsule, extended release - Oral, Kit, Tablet - Oral, Tablet, Tablet, film coated, extended release, Tablet, film coated, extended release - Oral, Intravenous, Injection, Injection - Intravenous, Tablet, film coated, Tablet, film coated - Oral, Powder, Powder - Oral, Capsule, coated pellets, Capsule, coated pellets - Oral, Topical, Aerosol, foam - Topical, Aerosol, foam
Rickettsia Infections
, 75.0 mg, 45.0 mg, 90.0 mg, 135.0 mg, 50.0 mg, 100.0 mg, 80.0 mg, 1.0 mg, 65.0 mg, 115.0 mg, 55.0 mg, 105.0 mg, 67.5 mg, 112.5 mg, 0.04 mg/mg, 0.015 mg/mg, 1.0 mg/mg
, Oral, Capsule - Oral, Capsule, Tablet, extended release, Tablet, extended release - Oral, Capsule, extended release, Capsule, extended release - Oral, Kit, Tablet - Oral, Tablet, Tablet, film coated, extended release, Tablet, film coated, extended release - Oral, Intravenous, Injection, Injection - Intravenous, Tablet, film coated, Tablet, film coated - Oral, Powder, Powder - Oral, Capsule, coated pellets, Capsule, coated pellets - Oral, Topical, Aerosol, foam - Topical, Aerosol, foam
Cat-Scratch Disease
, 75.0 mg, 45.0 mg, 90.0 mg, 135.0 mg, 50.0 mg, 100.0 mg, 80.0 mg, 1.0 mg, 65.0 mg, 115.0 mg, 55.0 mg, 105.0 mg, 67.5 mg, 112.5 mg, 0.04 mg/mg, 0.015 mg/mg, 1.0 mg/mg
, Oral, Capsule - Oral, Capsule, Tablet, extended release, Tablet, extended release - Oral, Capsule, extended release, Capsule, extended release - Oral, Kit, Tablet - Oral, Tablet, Tablet, film coated, extended release, Tablet, film coated, extended release - Oral, Intravenous, Injection, Injection - Intravenous, Tablet, film coated, Tablet, film coated - Oral, Powder, Powder - Oral, Capsule, coated pellets, Capsule, coated pellets - Oral, Topical, Aerosol, foam - Topical, Aerosol, foam
Dental Root Planing
, 75.0 mg, 45.0 mg, 90.0 mg, 135.0 mg, 50.0 mg, 100.0 mg, 80.0 mg, 1.0 mg, 65.0 mg, 115.0 mg, 55.0 mg, 105.0 mg, 67.5 mg, 112.5 mg, 0.04 mg/mg, 0.015 mg/mg, 1.0 mg/mg
, Oral, Capsule - Oral, Capsule, Tablet, extended release, Tablet, extended release - Oral, Capsule, extended release, Capsule, extended release - Oral, Kit, Tablet - Oral, Tablet, Tablet, film coated, extended release, Tablet, film coated, extended release - Oral, Intravenous, Injection, Injection - Intravenous, Tablet, film coated, Tablet, film coated - Oral, Powder, Powder - Oral, Capsule, coated pellets, Capsule, coated pellets - Oral, Topical, Aerosol, foam - Topical, Aerosol, foam
Plague
, 75.0 mg, 45.0 mg, 90.0 mg, 135.0 mg, 50.0 mg, 100.0 mg, 80.0 mg, 1.0 mg, 65.0 mg, 115.0 mg, 55.0 mg, 105.0 mg, 67.5 mg, 112.5 mg, 0.04 mg/mg, 0.015 mg/mg, 1.0 mg/mg
, Oral, Capsule - Oral, Capsule, Tablet, extended release, Tablet, extended release - Oral, Capsule, extended release, Capsule, extended release - Oral, Kit, Tablet - Oral, Tablet, Tablet, film coated, extended release, Tablet, film coated, extended release - Oral, Intravenous, Injection, Injection - Intravenous, Tablet, film coated, Tablet, film coated - Oral, Powder, Powder - Oral, Capsule, coated pellets, Capsule, coated pellets - Oral, Topical, Aerosol, foam - Topical, Aerosol, foam
Acne Vulgaris
, 75.0 mg, 45.0 mg, 90.0 mg, 135.0 mg, 50.0 mg, 100.0 mg, 80.0 mg, 1.0 mg, 65.0 mg, 115.0 mg, 55.0 mg, 105.0 mg, 67.5 mg, 112.5 mg, 0.04 mg/mg, 0.015 mg/mg, 1.0 mg/mg
, Oral, Capsule - Oral, Capsule, Tablet, extended release, Tablet, extended release - Oral, Capsule, extended release, Capsule, extended release - Oral, Kit, Tablet - Oral, Tablet, Tablet, film coated, extended release, Tablet, film coated, extended release - Oral, Intravenous, Injection, Injection - Intravenous, Tablet, film coated, Tablet, film coated - Oral, Powder, Powder - Oral, Capsule, coated pellets, Capsule, coated pellets - Oral, Topical, Aerosol, foam - Topical, Aerosol, foam
Rickettsialpox
, 75.0 mg, 45.0 mg, 90.0 mg, 135.0 mg, 50.0 mg, 100.0 mg, 80.0 mg, 1.0 mg, 65.0 mg, 115.0 mg, 55.0 mg, 105.0 mg, 67.5 mg, 112.5 mg, 0.04 mg/mg, 0.015 mg/mg, 1.0 mg/mg
, Oral, Capsule - Oral, Capsule, Tablet, extended release, Tablet, extended release - Oral, Capsule, extended release, Capsule, extended release - Oral, Kit, Tablet - Oral, Tablet, Tablet, film coated, extended release, Tablet, film coated, extended release - Oral, Intravenous, Injection, Injection - Intravenous, Tablet, film coated, Tablet, film coated - Oral, Powder, Powder - Oral, Capsule, coated pellets, Capsule, coated pellets - Oral, Topical, Aerosol, foam - Topical, Aerosol, foam
Disease
, 75.0 mg, 45.0 mg, 90.0 mg, 135.0 mg, 50.0 mg, 100.0 mg, 80.0 mg, 1.0 mg, 65.0 mg, 115.0 mg, 55.0 mg, 105.0 mg, 67.5 mg, 112.5 mg, 0.04 mg/mg, 0.015 mg/mg, 1.0 mg/mg
, Oral, Capsule - Oral, Capsule, Tablet, extended release, Tablet, extended release - Oral, Capsule, extended release, Capsule, extended release - Oral, Kit, Tablet - Oral, Tablet, Tablet, film coated, extended release, Tablet, film coated, extended release - Oral, Intravenous, Injection, Injection - Intravenous, Tablet, film coated, Tablet, film coated - Oral, Powder, Powder - Oral, Capsule, coated pellets, Capsule, coated pellets - Oral, Topical, Aerosol, foam - Topical, Aerosol, foam
Rocky Mountain Spotted Fever
, 75.0 mg, 45.0 mg, 90.0 mg, 135.0 mg, 50.0 mg, 100.0 mg, 80.0 mg, 1.0 mg, 65.0 mg, 115.0 mg, 55.0 mg, 105.0 mg, 67.5 mg, 112.5 mg, 0.04 mg/mg, 0.015 mg/mg, 1.0 mg/mg
, Oral, Capsule - Oral, Capsule, Tablet, extended release, Tablet, extended release - Oral, Capsule, extended release, Capsule, extended release - Oral, Kit, Tablet - Oral, Tablet, Tablet, film coated, extended release, Tablet, film coated, extended release - Oral, Intravenous, Injection, Injection - Intravenous, Tablet, film coated, Tablet, film coated - Oral, Powder, Powder - Oral, Capsule, coated pellets, Capsule, coated pellets - Oral, Topical, Aerosol, foam - Topical, Aerosol, foam
Relapsing Fever
, 75.0 mg, 45.0 mg, 90.0 mg, 135.0 mg, 50.0 mg, 100.0 mg, 80.0 mg, 1.0 mg, 65.0 mg, 115.0 mg, 55.0 mg, 105.0 mg, 67.5 mg, 112.5 mg, 0.04 mg/mg, 0.015 mg/mg, 1.0 mg/mg
, Oral, Capsule - Oral, Capsule, Tablet, extended release, Tablet, extended release - Oral, Capsule, extended release, Capsule, extended release - Oral, Kit, Tablet - Oral, Tablet, Tablet, film coated, extended release, Tablet, film coated, extended release - Oral, Intravenous, Injection, Injection - Intravenous, Tablet, film coated, Tablet, film coated - Oral, Powder, Powder - Oral, Capsule, coated pellets, Capsule, coated pellets - Oral, Topical, Aerosol, foam - Topical, Aerosol, foam
Trachoma
, 75.0 mg, 45.0 mg, 90.0 mg, 135.0 mg, 50.0 mg, 100.0 mg, 80.0 mg, 1.0 mg, 65.0 mg, 115.0 mg, 55.0 mg, 105.0 mg, 67.5 mg, 112.5 mg, 0.04 mg/mg, 0.015 mg/mg, 1.0 mg/mg
, Oral, Capsule - Oral, Capsule, Tablet, extended release, Tablet, extended release - Oral, Capsule, extended release, Capsule, extended release - Oral, Kit, Tablet - Oral, Tablet, Tablet, film coated, extended release, Tablet, film coated, extended release - Oral, Intravenous, Injection, Injection - Intravenous, Tablet, film coated, Tablet, film coated - Oral, Powder, Powder - Oral, Capsule, coated pellets, Capsule, coated pellets - Oral, Topical, Aerosol, foam - Topical, Aerosol, foam
Warnings
Arestin Contraindications
Condition
Risk Level
Notes
Pulse Frequency
Do Not Combine
Severe Hypersensitivity Reactions
Do Not Combine
Minocycline may interact with Pulse Frequency
There are 20 known major drug interactions with Arestin.
Common Arestin Drug Interactions
Drug Name
Risk Level
Description
Amdinocillin
Major
The therapeutic efficacy of Amdinocillin can be decreased when used in combination with Minocycline.
Amoxicillin
Major
The therapeutic efficacy of Amoxicillin can be decreased when used in combination with Minocycline.
Ampicillin
Major
The therapeutic efficacy of Ampicillin can be decreased when used in combination with Minocycline.
Aspoxicillin
Major
The therapeutic efficacy of Aspoxicillin can be decreased when used in combination with Minocycline.
Azidocillin
Major
The therapeutic efficacy of Azidocillin can be decreased when used in combination with Minocycline.
Arestin Toxicity & Overdose Risk
The lowest toxic dose of minocycline in rats is 2380mg/kg and 3600mg/kg in mice. The same dose in rats is 331mg/kg when administered through the abdomen and 1700mg/kg when given under the skin. A minocycline overdose may cause dizziness, nausea, and vomiting. Treatment involves stopping minocycline and providing symptom relief.
Arestin Novel Uses: Which Conditions Have a Clinical Trial Featuring Arestin?
There are currently 10 active studies investigating the potential of Arestin to alleviate Psittacosis, Tularemia and other Diseases.
Condition
Clinical Trials
Trial Phases
Gum Disease
3 Actively Recruiting
Phase 3, Not Applicable
Trachoma
2 Actively Recruiting
Phase 4, Not Applicable
Lymphogranuloma Venereum
0 Actively Recruiting
Disease
0 Actively Recruiting
Psittacosis
0 Actively Recruiting
Respiratory Tract Infections
0 Actively Recruiting
Dental Scaling
0 Actively Recruiting
Typhus, Endemic Flea-Borne
0 Actively Recruiting
Acne Vulgaris
0 Actively Recruiting
Relapsing Fever
0 Actively Recruiting
Plague
0 Actively Recruiting
Cat-Scratch Disease
0 Actively Recruiting
Rocky Mountain Spotted Fever
0 Actively Recruiting
Inflammation
0 Actively Recruiting
Brucellosis
0 Actively Recruiting
Rickettsia Infections
0 Actively Recruiting
Chancroid
0 Actively Recruiting
Q Fever
0 Actively Recruiting
Conjunctivitis, Inclusion
0 Actively Recruiting
Rickettsialpox
0 Actively Recruiting
Arestin Reviews: What are patients saying about Arestin?
5
Patient Review
12/14/2015
Arestin for Inflammation of the Tissues Surrounding a Tooth
4.3
Patient Review
11/16/2012
Arestin for Inflammation of the Tissues Surrounding a Tooth
2.7
Patient Review
1/24/2013
Arestin for Inflammation of the Tissues Surrounding a Tooth
2.3
Patient Review
5/4/2014
Arestin for Inflammation of the Tissues Surrounding a Tooth
2
Patient Review
7/16/2019
Arestin for Inflammation of the Tissues Surrounding a Tooth
1.7
Patient Review
2/26/2015
Arestin for Inflammation of the Tissues Surrounding a Tooth
1.7
Patient Review
11/2/2013
Arestin for Inflammation of the Tissues Surrounding a Tooth
1.3
Patient Review
9/23/2022
Arestin for Inflammation of the Tissues Surrounding a Tooth
1
Patient Review
11/11/2014
Arestin for Inflammation of the Tissues Surrounding a Tooth
1
Patient Review
3/11/2012
Arestin for Inflammation of the Tissues Surrounding a Tooth
1
Patient Review
8/22/2013
Arestin for Inflammation of the Tissues Surrounding a Tooth
1
Patient Review
4/15/2019
Arestin for Inflammation of the Tissues Surrounding a Tooth
Patient Q&A Section about arestin
These questions and answers are submitted by anonymous patients, and have not been verified by our internal team.
What is ARESTIN used for?
"ARESTIN® (minocycline HCl) Microspheres, 1mg is used in combination with Scaling and Root Planing (SRP) to treat patients with adult periodontitis (gum disease). ARESTIN® can be used as part of an overall oral health program that includes good brushing and flossing habits, as well as SRP."
Answered by AI
Is ARESTIN necessary?
"Medicating patients who don't need it is unnecessary for most patients as they typically respond well to non-surgical methods that don't involve antibiotics. This goes against the Centers for Disease Control (CDC) recommendations for appropriate antibiotic use."
Answered by AI
What is a dental ARESTIN?
"Arestin is a dental antibiotic which is placed directly into infected gum pockets by a professional after a scaling and root planing procedure. Arestin is more effective than root planing alone in fighting against harmful bacteria."
Answered by AI
How long does ARESTIN last for?
"Arestin starts working quickly, right at the source of infection and keeps fighting bacteria long after you leave the dental office. Arestin fights infection and inflammation for 30 days and provides significantly better results than scaling and root planing alone for up to 90 days."
Answered by AI