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What is Omeprazole Magnesium
EsomeprazoleThe Generic name of this drug
Treatment SummaryEsomeprazole, sold under the brand name Nexium, is a medication used to treat gastroesophageal reflux disease (GERD), peptic ulcer disease, and other disorders related to too much stomach acid. It is a proton pump inhibitor (PPI) and works by blocking the production of stomach acid. Esomeprazole is usually prescribed with other antibiotics to help treat _H. pylori_ infections. It is generally safe and effective, but long-term use can lead to some side effects such as an increased risk of bacterial infections and reduced absorption of certain vitamins and minerals. Rapid
Nexiumis the brand name
Omeprazole Magnesium Overview & Background
Brand Name
Generic Name
First FDA Approval
How many FDA approvals?
Nexium
Esomeprazole
2001
347
Approved as Treatment by the FDA
Esomeprazole, otherwise called Nexium, is approved by the FDA for 3 uses including Heartburn and Heartburn .Heartburn
Heartburn
Helps manage Gastro-esophageal Reflux Disease (GERD)
Helicobacter Pylori Infection
Used to treat Helicobacter Pylori Infection in combination with Amoxicillin
Effectiveness
How Omeprazole Magnesium Affects PatientsEsomeprazole is a drug that stops stomach acid from being released. It is used to treat GERD, heal damage to the esophagus, and to prevent ulcers in the stomach. It works by blocking the enzyme (H+/K+ ATPase) on the stomach wall that is responsible for producing acid. Esomeprazole is similar to another antacid, [DB00338], but does not have the same side effects. Taking esomeprazole long-term can lead to some risks, including increased risk of bacterial infections, difficulty absorbing certain vitamins, low magnesium levels, and
How Omeprazole Magnesium works in the bodyEsomeprazole works by blocking the enzyme that produces stomach acid. This enzyme, called the (H+, K+)-ATPase, is found on the surface of stomach cells. When esomeprazole binds to it, it stops the enzyme from creating acid. This effect lasts longer than 24 hours, and new enzyme needs to be produced for acid production to resume.
When to interrupt dosage
The suggested dosage of Omeprazole Magnesium is contingent upon the diagnosed condition, including Curling Ulcer, Hemorrhage and Critical Illness. The quantity of dosage fluctuates as per the approach of administration (e.g. Tablet, delayed release or Injection, powder, lyophilized, for solution - Intravenous) outlined in the table beneath.Condition
Dosage
Administration
Heartburn
20.0 mg, , 40.0 mg, 20.0 mg/mL, 40.0 mg/mL, 10.0 mg, 2.5 mg, 5.0 mg, 24.65 mg, 49.3 mg
, Capsule, delayed release, Oral, Capsule, delayed release - Oral, Tablet, delayed release, Tablet, delayed release - Oral, Intravenous, Injection, powder, lyophilized, for solution, Injection, powder, lyophilized, for solution - Intravenous, Granule, delayed release, Granule, delayed release - Oral, Injection, Injection - Intravenous, Capsule, delayed release pellets, Capsule, delayed release pellets - Oral, Tablet, Tablet - Oral, Kit, Capsule, Capsule - Oral, Granule, for suspension, extended release, For suspension - Oral, For suspension, Granule, for suspension, extended release - Oral, Capsule, coated pellets, Kit - Oral, Capsule, coated pellets - Oral, Tablet, film coated - Oral, Tablet, film coated
Hemorrhage
20.0 mg, , 40.0 mg, 20.0 mg/mL, 40.0 mg/mL, 10.0 mg, 2.5 mg, 5.0 mg, 24.65 mg, 49.3 mg
, Capsule, delayed release, Oral, Capsule, delayed release - Oral, Tablet, delayed release, Tablet, delayed release - Oral, Intravenous, Injection, powder, lyophilized, for solution, Injection, powder, lyophilized, for solution - Intravenous, Granule, delayed release, Granule, delayed release - Oral, Injection, Injection - Intravenous, Capsule, delayed release pellets, Capsule, delayed release pellets - Oral, Tablet, Tablet - Oral, Kit, Capsule, Capsule - Oral, Granule, for suspension, extended release, For suspension - Oral, For suspension, Granule, for suspension, extended release - Oral, Capsule, coated pellets, Kit - Oral, Capsule, coated pellets - Oral, Tablet, film coated - Oral, Tablet, film coated
maintenance of healing Erosive esophagitis
20.0 mg, , 40.0 mg, 20.0 mg/mL, 40.0 mg/mL, 10.0 mg, 2.5 mg, 5.0 mg, 24.65 mg, 49.3 mg
, Capsule, delayed release, Oral, Capsule, delayed release - Oral, Tablet, delayed release, Tablet, delayed release - Oral, Intravenous, Injection, powder, lyophilized, for solution, Injection, powder, lyophilized, for solution - Intravenous, Granule, delayed release, Granule, delayed release - Oral, Injection, Injection - Intravenous, Capsule, delayed release pellets, Capsule, delayed release pellets - Oral, Tablet, Tablet - Oral, Kit, Capsule, Capsule - Oral, Granule, for suspension, extended release, For suspension - Oral, For suspension, Granule, for suspension, extended release - Oral, Capsule, coated pellets, Kit - Oral, Capsule, coated pellets - Oral, Tablet, film coated - Oral, Tablet, film coated
Peptic Ulcer
20.0 mg, , 40.0 mg, 20.0 mg/mL, 40.0 mg/mL, 10.0 mg, 2.5 mg, 5.0 mg, 24.65 mg, 49.3 mg
, Capsule, delayed release, Oral, Capsule, delayed release - Oral, Tablet, delayed release, Tablet, delayed release - Oral, Intravenous, Injection, powder, lyophilized, for solution, Injection, powder, lyophilized, for solution - Intravenous, Granule, delayed release, Granule, delayed release - Oral, Injection, Injection - Intravenous, Capsule, delayed release pellets, Capsule, delayed release pellets - Oral, Tablet, Tablet - Oral, Kit, Capsule, Capsule - Oral, Granule, for suspension, extended release, For suspension - Oral, For suspension, Granule, for suspension, extended release - Oral, Capsule, coated pellets, Kit - Oral, Capsule, coated pellets - Oral, Tablet, film coated - Oral, Tablet, film coated
Critical Illness
20.0 mg, , 40.0 mg, 20.0 mg/mL, 40.0 mg/mL, 10.0 mg, 2.5 mg, 5.0 mg, 24.65 mg, 49.3 mg
, Capsule, delayed release, Oral, Capsule, delayed release - Oral, Tablet, delayed release, Tablet, delayed release - Oral, Intravenous, Injection, powder, lyophilized, for solution, Injection, powder, lyophilized, for solution - Intravenous, Granule, delayed release, Granule, delayed release - Oral, Injection, Injection - Intravenous, Capsule, delayed release pellets, Capsule, delayed release pellets - Oral, Tablet, Tablet - Oral, Kit, Capsule, Capsule - Oral, Granule, for suspension, extended release, For suspension - Oral, For suspension, Granule, for suspension, extended release - Oral, Capsule, coated pellets, Kit - Oral, Capsule, coated pellets - Oral, Tablet, film coated - Oral, Tablet, film coated
Stress Ulcers
20.0 mg, , 40.0 mg, 20.0 mg/mL, 40.0 mg/mL, 10.0 mg, 2.5 mg, 5.0 mg, 24.65 mg, 49.3 mg
, Capsule, delayed release, Oral, Capsule, delayed release - Oral, Tablet, delayed release, Tablet, delayed release - Oral, Intravenous, Injection, powder, lyophilized, for solution, Injection, powder, lyophilized, for solution - Intravenous, Granule, delayed release, Granule, delayed release - Oral, Injection, Injection - Intravenous, Capsule, delayed release pellets, Capsule, delayed release pellets - Oral, Tablet, Tablet - Oral, Kit, Capsule, Capsule - Oral, Granule, for suspension, extended release, For suspension - Oral, For suspension, Granule, for suspension, extended release - Oral, Capsule, coated pellets, Kit - Oral, Capsule, coated pellets - Oral, Tablet, film coated - Oral, Tablet, film coated
previous gastric or duodenal ulcer
20.0 mg, , 40.0 mg, 20.0 mg/mL, 40.0 mg/mL, 10.0 mg, 2.5 mg, 5.0 mg, 24.65 mg, 49.3 mg
, Capsule, delayed release, Oral, Capsule, delayed release - Oral, Tablet, delayed release, Tablet, delayed release - Oral, Intravenous, Injection, powder, lyophilized, for solution, Injection, powder, lyophilized, for solution - Intravenous, Granule, delayed release, Granule, delayed release - Oral, Injection, Injection - Intravenous, Capsule, delayed release pellets, Capsule, delayed release pellets - Oral, Tablet, Tablet - Oral, Kit, Capsule, Capsule - Oral, Granule, for suspension, extended release, For suspension - Oral, For suspension, Granule, for suspension, extended release - Oral, Capsule, coated pellets, Kit - Oral, Capsule, coated pellets - Oral, Tablet, film coated - Oral, Tablet, film coated
antibacterial therapy
20.0 mg, , 40.0 mg, 20.0 mg/mL, 40.0 mg/mL, 10.0 mg, 2.5 mg, 5.0 mg, 24.65 mg, 49.3 mg
, Capsule, delayed release, Oral, Capsule, delayed release - Oral, Tablet, delayed release, Tablet, delayed release - Oral, Intravenous, Injection, powder, lyophilized, for solution, Injection, powder, lyophilized, for solution - Intravenous, Granule, delayed release, Granule, delayed release - Oral, Injection, Injection - Intravenous, Capsule, delayed release pellets, Capsule, delayed release pellets - Oral, Tablet, Tablet - Oral, Kit, Capsule, Capsule - Oral, Granule, for suspension, extended release, For suspension - Oral, For suspension, Granule, for suspension, extended release - Oral, Capsule, coated pellets, Kit - Oral, Capsule, coated pellets - Oral, Tablet, film coated - Oral, Tablet, film coated
Heartburn
20.0 mg, , 40.0 mg, 20.0 mg/mL, 40.0 mg/mL, 10.0 mg, 2.5 mg, 5.0 mg, 24.65 mg, 49.3 mg
, Capsule, delayed release, Oral, Capsule, delayed release - Oral, Tablet, delayed release, Tablet, delayed release - Oral, Intravenous, Injection, powder, lyophilized, for solution, Injection, powder, lyophilized, for solution - Intravenous, Granule, delayed release, Granule, delayed release - Oral, Injection, Injection - Intravenous, Capsule, delayed release pellets, Capsule, delayed release pellets - Oral, Tablet, Tablet - Oral, Kit, Capsule, Capsule - Oral, Granule, for suspension, extended release, For suspension - Oral, For suspension, Granule, for suspension, extended release - Oral, Capsule, coated pellets, Kit - Oral, Capsule, coated pellets - Oral, Tablet, film coated - Oral, Tablet, film coated
develop NSAID-induced gastric ulcers
20.0 mg, , 40.0 mg, 20.0 mg/mL, 40.0 mg/mL, 10.0 mg, 2.5 mg, 5.0 mg, 24.65 mg, 49.3 mg
, Capsule, delayed release, Oral, Capsule, delayed release - Oral, Tablet, delayed release, Tablet, delayed release - Oral, Intravenous, Injection, powder, lyophilized, for solution, Injection, powder, lyophilized, for solution - Intravenous, Granule, delayed release, Granule, delayed release - Oral, Injection, Injection - Intravenous, Capsule, delayed release pellets, Capsule, delayed release pellets - Oral, Tablet, Tablet - Oral, Kit, Capsule, Capsule - Oral, Granule, for suspension, extended release, For suspension - Oral, For suspension, Granule, for suspension, extended release - Oral, Capsule, coated pellets, Kit - Oral, Capsule, coated pellets - Oral, Tablet, film coated - Oral, Tablet, film coated
Helicobacter Pylori Infection
20.0 mg, , 40.0 mg, 20.0 mg/mL, 40.0 mg/mL, 10.0 mg, 2.5 mg, 5.0 mg, 24.65 mg, 49.3 mg
, Capsule, delayed release, Oral, Capsule, delayed release - Oral, Tablet, delayed release, Tablet, delayed release - Oral, Intravenous, Injection, powder, lyophilized, for solution, Injection, powder, lyophilized, for solution - Intravenous, Granule, delayed release, Granule, delayed release - Oral, Injection, Injection - Intravenous, Capsule, delayed release pellets, Capsule, delayed release pellets - Oral, Tablet, Tablet - Oral, Kit, Capsule, Capsule - Oral, Granule, for suspension, extended release, For suspension - Oral, For suspension, Granule, for suspension, extended release - Oral, Capsule, coated pellets, Kit - Oral, Capsule, coated pellets - Oral, Tablet, film coated - Oral, Tablet, film coated
Hemorrhage
20.0 mg, , 40.0 mg, 20.0 mg/mL, 40.0 mg/mL, 10.0 mg, 2.5 mg, 5.0 mg, 24.65 mg, 49.3 mg
, Capsule, delayed release, Oral, Capsule, delayed release - Oral, Tablet, delayed release, Tablet, delayed release - Oral, Intravenous, Injection, powder, lyophilized, for solution, Injection, powder, lyophilized, for solution - Intravenous, Granule, delayed release, Granule, delayed release - Oral, Injection, Injection - Intravenous, Capsule, delayed release pellets, Capsule, delayed release pellets - Oral, Tablet, Tablet - Oral, Kit, Capsule, Capsule - Oral, Granule, for suspension, extended release, For suspension - Oral, For suspension, Granule, for suspension, extended release - Oral, Capsule, coated pellets, Kit - Oral, Capsule, coated pellets - Oral, Tablet, film coated - Oral, Tablet, film coated
Erosive Esophagitis
20.0 mg, , 40.0 mg, 20.0 mg/mL, 40.0 mg/mL, 10.0 mg, 2.5 mg, 5.0 mg, 24.65 mg, 49.3 mg
, Capsule, delayed release, Oral, Capsule, delayed release - Oral, Tablet, delayed release, Tablet, delayed release - Oral, Intravenous, Injection, powder, lyophilized, for solution, Injection, powder, lyophilized, for solution - Intravenous, Granule, delayed release, Granule, delayed release - Oral, Injection, Injection - Intravenous, Capsule, delayed release pellets, Capsule, delayed release pellets - Oral, Tablet, Tablet - Oral, Kit, Capsule, Capsule - Oral, Granule, for suspension, extended release, For suspension - Oral, For suspension, Granule, for suspension, extended release - Oral, Capsule, coated pellets, Kit - Oral, Capsule, coated pellets - Oral, Tablet, film coated - Oral, Tablet, film coated
Gastric ulcer
20.0 mg, , 40.0 mg, 20.0 mg/mL, 40.0 mg/mL, 10.0 mg, 2.5 mg, 5.0 mg, 24.65 mg, 49.3 mg
, Capsule, delayed release, Oral, Capsule, delayed release - Oral, Tablet, delayed release, Tablet, delayed release - Oral, Intravenous, Injection, powder, lyophilized, for solution, Injection, powder, lyophilized, for solution - Intravenous, Granule, delayed release, Granule, delayed release - Oral, Injection, Injection - Intravenous, Capsule, delayed release pellets, Capsule, delayed release pellets - Oral, Tablet, Tablet - Oral, Kit, Capsule, Capsule - Oral, Granule, for suspension, extended release, For suspension - Oral, For suspension, Granule, for suspension, extended release - Oral, Capsule, coated pellets, Kit - Oral, Capsule, coated pellets - Oral, Tablet, film coated - Oral, Tablet, film coated
prophylaxis of Stress Ulcers
20.0 mg, , 40.0 mg, 20.0 mg/mL, 40.0 mg/mL, 10.0 mg, 2.5 mg, 5.0 mg, 24.65 mg, 49.3 mg
, Capsule, delayed release, Oral, Capsule, delayed release - Oral, Tablet, delayed release, Tablet, delayed release - Oral, Intravenous, Injection, powder, lyophilized, for solution, Injection, powder, lyophilized, for solution - Intravenous, Granule, delayed release, Granule, delayed release - Oral, Injection, Injection - Intravenous, Capsule, delayed release pellets, Capsule, delayed release pellets - Oral, Tablet, Tablet - Oral, Kit, Capsule, Capsule - Oral, Granule, for suspension, extended release, For suspension - Oral, For suspension, Granule, for suspension, extended release - Oral, Capsule, coated pellets, Kit - Oral, Capsule, coated pellets - Oral, Tablet, film coated - Oral, Tablet, film coated
Zollinger-Ellison Syndrome
20.0 mg, , 40.0 mg, 20.0 mg/mL, 40.0 mg/mL, 10.0 mg, 2.5 mg, 5.0 mg, 24.65 mg, 49.3 mg
, Capsule, delayed release, Oral, Capsule, delayed release - Oral, Tablet, delayed release, Tablet, delayed release - Oral, Intravenous, Injection, powder, lyophilized, for solution, Injection, powder, lyophilized, for solution - Intravenous, Granule, delayed release, Granule, delayed release - Oral, Injection, Injection - Intravenous, Capsule, delayed release pellets, Capsule, delayed release pellets - Oral, Tablet, Tablet - Oral, Kit, Capsule, Capsule - Oral, Granule, for suspension, extended release, For suspension - Oral, For suspension, Granule, for suspension, extended release - Oral, Capsule, coated pellets, Kit - Oral, Capsule, coated pellets - Oral, Tablet, film coated - Oral, Tablet, film coated
Curling Ulcer
20.0 mg, , 40.0 mg, 20.0 mg/mL, 40.0 mg/mL, 10.0 mg, 2.5 mg, 5.0 mg, 24.65 mg, 49.3 mg
, Capsule, delayed release, Oral, Capsule, delayed release - Oral, Tablet, delayed release, Tablet, delayed release - Oral, Intravenous, Injection, powder, lyophilized, for solution, Injection, powder, lyophilized, for solution - Intravenous, Granule, delayed release, Granule, delayed release - Oral, Injection, Injection - Intravenous, Capsule, delayed release pellets, Capsule, delayed release pellets - Oral, Tablet, Tablet - Oral, Kit, Capsule, Capsule - Oral, Granule, for suspension, extended release, For suspension - Oral, For suspension, Granule, for suspension, extended release - Oral, Capsule, coated pellets, Kit - Oral, Capsule, coated pellets - Oral, Tablet, film coated - Oral, Tablet, film coated
Warnings
Omeprazole Magnesium has a single contraindication and should not be employed when one is suffering from any of the conditions outlined in the table below.Omeprazole Magnesium ContraindicationsCondition
Risk Level
Notes
Pulse Frequency
Do Not Combine
Common Omeprazole Magnesium Drug Interactions
Drug Name
Risk Level
Description
Acenocoumarol
Major
The metabolism of Acenocoumarol can be decreased when combined with Esomeprazole.
Atazanavir
Major
Esomeprazole can cause a decrease in the absorption of Atazanavir resulting in a reduced serum concentration and potentially a decrease in efficacy.
Axitinib
Major
The metabolism of Axitinib can be decreased when combined with Esomeprazole.
Cyclophosphamide
Major
The metabolism of Cyclophosphamide can be decreased when combined with Esomeprazole.
Infigratinib
Major
The serum concentration of Infigratinib can be decreased when it is combined with Esomeprazole.
Omeprazole Magnesium Toxicity & Overdose RiskTaking too much of this drug may cause blurry vision, confusion, drowsiness, thirst, redness in the face, headache, stomach upset, an unusually fast heart rate, and excessive sweating.
Omeprazole Magnesium Novel Uses: Which Conditions Have a Clinical Trial Featuring Omeprazole Magnesium?
Currently, 26 active trials are examining the potential of Omeprazole Magnesium in treating prior gastric or duodenal ulcer, Stomach Ulcer and Peptic Ulcer Disorders.Condition
Clinical Trials
Trial Phases
Heartburn
2 Actively Recruiting
Phase 3, Not Applicable
Helicobacter Pylori Infection
0 Actively Recruiting
Curling Ulcer
0 Actively Recruiting
previous gastric or duodenal ulcer
0 Actively Recruiting
Zollinger-Ellison Syndrome
0 Actively Recruiting
antibacterial therapy
0 Actively Recruiting
develop NSAID-induced gastric ulcers
0 Actively Recruiting
Peptic Ulcer
2 Actively Recruiting
Not Applicable, Phase 4
Hemorrhage
1 Actively Recruiting
Phase 4
Gastric ulcer
0 Actively Recruiting
Erosive Esophagitis
3 Actively Recruiting
Phase 2, Phase 3
maintenance of healing Erosive esophagitis
0 Actively Recruiting
Heartburn
14 Actively Recruiting
Phase 3, Phase 2, Not Applicable, Phase 4, Phase 1
Hemorrhage
0 Actively Recruiting
prophylaxis of Stress Ulcers
0 Actively Recruiting
Stress Ulcers
0 Actively Recruiting
Critical Illness
0 Actively Recruiting
Omeprazole Magnesium Reviews: What are patients saying about Omeprazole Magnesium?
5Patient Review
8/23/2013 I was taking one 20ml tablet a day and it didn't seem to be doing much. I then started taking two pills each day, one in the morning and one at night. However, after a couple of weeks on this higher dosage, I started experiencing some pain on the left side of my back. Once I stopped taking the pills, the pain went away.
5Patient Review
12/25/2013 I take this medication first thing in the morning and it really does help reduce or eliminate my heartburn symptoms. I've been taking it for years and would recommend it to others.
5Patient Review
3/16/20115Patient Review
11/20/20115Patient Review
4/18/2013 I've been on a lot of different medications for my heartburn, and none of them have really worked. I'm disappointed that after two years, I'm still not any better.
5Patient Review
1/15/2017 Though it doesn't work in the same way as Nexium, this drug was highly effective for me. I really enjoyed taking it!
4.7Patient Review
7/28/20114.7Patient Review
6/11/20124.7Patient Review
7/28/2014 This medication is very effective and very affordable.
4.3Patient Review
6/6/2018 This medication has been a total game-changer for me and my acid reflux. I never forget to take it because it's such an easy pill to remember, and since starting it I haven't had any issues at all.
4.3Patient Review
2/16/2020 I've used this for 12 years and, for a long time, still battled with reflux. I finally discovered that the key is to take a lower dose than what is typically prescribed. Now, I haven't had any problems in over two years.
3.7Patient Review
10/4/2012 I was taking anti-inflammatory drugs but developed stomach pains. This medication worked well for me.
3.7Patient Review
10/25/2016 The medication worked but after taking it for just over a year, I started having hand tremors Went thru tests, including an MRI. After renewing my prescription, I read the insert more carefully. Seems it lowers the magnesium levels, which caused my problem, plus heart palpatations, rashes, & more. I've stopped the medication & will start Mg supplementation.
3.7Patient Review
4/28/2013 I've taken omeprazole before and found it very easy to use. I didn't experience any negative effects, even after using it for more than two weeks straight.
3.7Patient Review
4/6/20113.3Patient Review
2/2/2015 I wonder how this medication will affect the absorption of methotrexate. I noticed that on this site, it says that methotrexate is a drug with interactions?
1Patient Review
1/3/2013 While this medication was successful in reducing stomach acid, I began experiencing anxiety, tachycardia, and hypertension. After getting a full cardiac workup (which came back negative), I stopped taking the drug and my symptoms immediately disappeared.
1Patient Review
4/23/2012Patient Q&A Section about omeprazole magnesium
These questions and answers are submitted by anonymous patients, and have not been verified by our internal team.Does omeprazole cause low magnesium?
"The majority of reports of low magnesium levels have been linked to extended use of omeprazole at standard doses (20-40mg daily). after discontinuing the medication, magnesium levels returned to normal."
Answered by AI
Is omeprazole the same as omeprazole magnesium?
"Omeprazole Magnesium is a generic drug, also known by its brand name, First-Omeprazole."
Answered by AI
Does magnesium interact with omeprazole?
"There are no known interactions between Chelated Magnesium and omeprazole, but this does not mean that interactions can't exist. Always check with your healthcare provider."
Answered by AI
What does omeprazole magnesium do?
"This medication works by decreasing the amount of acid your stomach makes, relieving symptoms such as heartburn, difficulty swallowing, and cough. It also helps heal acid damage to the stomach and esophagus, helps prevent ulcers, and may help prevent cancer of the esophagus."
Answered by AI