Decitabine + Cedazuridine + Enzalutamide for Prostate Cancer

Age: 18+
Sex: Male
Trial Phase: Phase 1
Sponsor: Roswell Park Cancer Institute
Must be taking: Enzalutamide
No Placebo GroupAll trial participants will receive the active study treatment (no placebo)

What You Need to Know Before You Apply

What is the purpose of this trial?

This trial tests a combination of medications to determine the optimal dose and effects for treating prostate cancer that has spread and resists standard hormonal treatments. It examines the use of decitabine/cedazuridine (a combination drug) with enzalutamide (a hormonal therapy) to overcome the cancer's resistance to enzalutamide alone. Men with prostate cancer that no longer responds to usual treatments and is spreading might be suitable candidates, especially if they currently take enzalutamide. As a Phase 1 trial, the research aims to understand how the treatment works in people, offering participants the chance to be among the first to receive this new combination therapy.

Do I have to stop taking my current medications for the trial?

You may need to stop taking certain medications, especially if they are strong inducers or inhibitors of CYP3A4/5, at least 7 days before starting the trial. It's best to discuss your current medications with the trial team to see if any adjustments are needed.

Is there any evidence suggesting that this trial's treatments are likely to be safe?

Research has shown that combining decitabine and cedazuridine is generally as safe as other similar treatments, meaning most people tolerate them well. Some side effects may occur, but they are typical for chemotherapy drugs. Studies indicate that enzalutamide can lower the risk of death in prostate cancer patients. It is usually safe, though it may cause some side effects, like most medications.

Overall, both treatments are considered manageable in terms of safety, with careful monitoring advised. Prospective trial participants should discuss these findings with their doctor to make an informed decision.12345

Why are researchers excited about this study treatment for prostate cancer?

Researchers are excited about the combination of decitabine, cedazuridine, and enzalutamide for prostate cancer because it offers a novel approach by combining epigenetic modification with hormone therapy. Decitabine and cedazuridine work together to inhibit DNA methylation, potentially reactivating genes that suppress tumor growth, while enzalutamide targets androgen receptors to block the effects of male hormones that can fuel cancer. This dual-action strategy could enhance the effectiveness of prostate cancer treatment, offering hope for better outcomes compared to the current standard of care, which typically focuses on hormone therapy alone.

What evidence suggests that this trial's treatments could be effective for prostate cancer?

Studies have shown that enzalutamide can significantly improve survival for prostate cancer patients. Specifically, men taking enzalutamide had a 61% lower chance of their cancer worsening compared to those not taking it. Other research found that enzalutamide reduced the risk of death by 33% compared to a group not receiving the treatment. The combination of decitabine and cedazuridine has also shown promise, with patients having certain blood cancers living a median of 31.7 months. In this trial, participants will receive both enzalutamide and the combination of decitabine and cedazuridine. Together, these treatments might help overcome resistance to enzalutamide alone, potentially offering a new way to manage advanced prostate cancer.16789

Who Is on the Research Team?

Gurkamal Chatta MD | Roswell Park ...

Gurkamal Chatta, Dr.

Principal Investigator

Roswell Park Cancer Institute

Are You a Good Fit for This Trial?

Men over 18 with metastatic castrate resistant prostate cancer, showing disease progression. They must have good performance status (able to carry out daily activities), low testosterone levels if not on androgen deprivation therapy, adequate organ function, and the ability to swallow pills. Prior treatments for prostate cancer are allowed in some phases of the trial. Participants must use contraception.

Inclusion Criteria

I can swallow and keep down pills.
I am fully active or can carry out light work.
Understanding and signing an informed consent form
See 5 more

Exclusion Criteria

I haven't had another cancer within the last 3 years.
Unsuitable candidate to receive study drug
I am taking certain medications that I cannot stop.
See 8 more

Timeline for a Trial Participant

Screening

Participants are screened for eligibility to participate in the trial

2-4 weeks

Treatment

Participants receive decitabine and cedazuridine orally once daily on either days 1-3, 1-4, or 1-5 and enzalutamide orally once daily on days 1-28. Treatments repeat every 28 days for up to 6 cycles.

24 weeks

Follow-up

Participants are monitored for safety and effectiveness after treatment completion

24 months
Follow-up at 30 days, then every 3 months

What Are the Treatments Tested in This Trial?

Interventions

  • Decitabine and Cedazuridine
  • Enzalutamide
Trial Overview The trial is testing the combination of decitabine/cedazuridine with enzalutamide to determine safe dosages and potential benefits or side effects in treating advanced prostate cancer that resists standard treatment. The goal is also to see if this combo can overcome resistance developed against enzalutamide alone.
How Is the Trial Designed?
1Treatment groups
Experimental Treatment
Group I: Treatment (decitabine and cedazuridine, enzalutamide)Experimental Treatment2 Interventions

Decitabine and Cedazuridine is already approved in European Union, United States for the following indications:

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Approved in European Union as Inaqovi for:
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Approved in United States as ASTX727 for:

Find a Clinic Near You

Who Is Running the Clinical Trial?

Roswell Park Cancer Institute

Lead Sponsor

Trials
427
Recruited
40,500+

National Comprehensive Cancer Network

Collaborator

Trials
121
Recruited
7,400+

Citations

Correlative results from NCI CTEP/ETCTN 10330: A phase ...Results: 19 pts were treated; all received paired biopsies. WES was adequate in 7/19 (37%) pts, with IDHm identified in 3/7 (43%) pts. All pts ...
Study Details | NCT05037500 | Decitabine/Cedazuridine ...This phase Ib trial is to find out the best dose decitabine/cedazuridine and possible benefits and/or side effects of decitabine/cedazuridine and ...
Phase 2 Study of Oral Decitabine/Cedazuridine in ...To evaluate preliminary safety and efficacy of oral decitabine/cedazuridine in combination with magrolimab. Primary Objective. •To evaluate the ...
Prolonged Overall Survival Observed With Oral Decitabine ...The oral, fixed-duration combination of decitabine and cedazuridine induced a median overall survival of 31.7 months in patients with intermediate- and high- ...
FDA Accepts sNDA for Decitabine/Cedazuridine Combo in ...The CR rate was 46.5% (95% CI, 36.5%-56.7%), with a CRi rate of 16.8%, CRh rate of 5.0%, a CR plus CRi rate of 63.4% (95% CI, 53.2%-72.7%), a CR ...
Phase II trial of 10-day ASTX727 (decitabine/cedazuridine ...Conclusions: The 10-day ASTX727-VEN combination showed safety profile comparable to other HMA-VEN regimens in salvage setting. ... Outcomes of 10- ...
Highlights of the NCCN Oncology Research Program inGiving decitabine/cedazuridine together with enzalutamide may reverse or help prevent the acquired therapeutic resistance that is observed when ...
ASTX029 and Decitabine and Cedazuridine (ASTX727) for ...Cedazuridine helps decitabine work better by helping to prevent its breakdown in the body. Giving ASTX029 and ASTX727 may be a safe and effective treatment ...
Astex Pharmaceuticals, Inc. ASTX727 Clinical ProtocolBased on this outcome, a dose combination of 100 mg cedazuridine with 35 mg decitabine (ie, intermediate dose between 30 mg and 40 mg) was selected for the ...
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