250 Participants Needed

MK-4716 for Cancer

Recruiting at 1 trial location
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No Placebo GroupAll trial participants will receive the active study treatment (no placebo)

What You Need to Know Before You Apply

What is the purpose of this trial?

This trial explores a new treatment called MK-4716 for certain advanced or metastatic cancers. Researchers aim to assess the safety of MK-4716 and its tolerability, both alone and in combination with other treatments like Pembrolizumab and Cetuximab. The trial seeks participants with specific types of solid tumors, such as advanced lung cancer or tumors with a KRAS gene change, who have undergone previous treatments. Participants should have measurable disease and be able to swallow pills. As a Phase 1 trial, this research focuses on understanding how MK-4716 works in people, offering participants the opportunity to be among the first to receive this new treatment.

Will I have to stop taking my current medications?

The trial information does not specify if you need to stop taking your current medications. However, if you are on immunosuppressive therapy or have received prior immunotherapy, you may not be eligible for certain parts of the trial.

Is there any evidence suggesting that this trial's treatments are likely to be safe?

A previous study on MK-4716 focused on its safety when used alone or with other treatments. When combined with pembrolizumab, the drug showed a manageable safety profile. Most side effects were mild or moderate, such as tiredness or nausea. Pembrolizumab, already used for other cancers, typically causes mild side effects, which are well-known and manageable.

For MK-4716 combined with cetuximab, cetuximab is approved for some cancers and usually causes side effects like skin reactions and low magnesium levels. These are common and treatable.

Since MK-4716 is in an early trial phase, the main goal is to test its safety. At this stage, researchers aim to find the right dose and check for any side effects, but clear data on MK-4716 alone remains limited. This trial is crucial to ensure the treatment is safe and tolerable.12345

Why are researchers excited about this trial's treatments?

Researchers are excited about MK-4716 for cancer because it offers a unique approach compared to standard treatments like chemotherapy and targeted therapies. Unlike most treatments that attack cancer cells directly, MK-4716 may work by enhancing the body's immune response to target cancer cells more effectively. Additionally, when combined with drugs like Pembrolizumab or Cetuximab, MK-4716 has the potential to improve the effectiveness of these existing immunotherapy and targeted therapy options, potentially leading to better outcomes for patients. This new mechanism and combination strategy represent a promising step forward in cancer treatment.

What evidence suggests that MK-4716 could be an effective treatment for advanced or metastatic solid tumors?

Studies have shown that researchers are investigating MK-4716 for its potential to treat certain advanced cancers. This drug targets specific cancer pathways, which may stop tumors from growing. In this trial, participants will receive MK-4716 in different treatment arms. One arm involves MK-4716 alone at varying dose levels and schedules. Another arm combines MK-4716 with pembrolizumab, a drug that helps the immune system fight cancer and has shown some success in treating lung cancer. Researchers are also exploring a combination of MK-4716 with cetuximab, which has been helpful for some colorectal cancers. Although much remains to be learned, these early results offer promise for people with difficult-to-treat tumors.16789

Who Is on the Research Team?

MD

Medical Director

Principal Investigator

Merck Sharp & Dohme LLC

Are You a Good Fit for This Trial?

This trial is for people with certain advanced solid tumors who've had at least one systemic therapy. Specifically, it's for those with a confirmed diagnosis of unresectable or metastatic solid tumors or non-small cell lung cancer that have KRAS alterations. Participants must be able to swallow pills and haven't been treated yet if they have lung cancer.

Inclusion Criteria

I have had at least one treatment for my advanced cancer that cannot be surgically removed.
I have been diagnosed with metastatic non-small cell lung cancer.
My cancer has a KRAS mutation.
See 5 more

Timeline for a Trial Participant

Screening

Participants are screened for eligibility to participate in the trial

2-4 weeks

Treatment

Participants receive MK-4716 as monotherapy or in combination with Pembrolizumab or Cetuximab

8 weeks

Follow-up

Participants are monitored for safety and effectiveness after treatment

5 years

Pharmacokinetics Assessment

Blood samples are collected to determine pharmacokinetic parameters such as AUC, Cmax, and Ctrough of MK-4716

58 days

What Are the Treatments Tested in This Trial?

Interventions

  • MK-4716

Trial Overview

The study is testing the safety and tolerance of MK-4716 alone or combined with Cetuximab or Pembrolizumab in treating advanced cancers. It aims to find out how well these treatments work on specific solid tumors, including those with genetic changes like KRAS mutations.

How Is the Trial Designed?

3

Treatment groups

Experimental Treatment

Group I: MK-4716 Dose EscalationExperimental Treatment1 Intervention
Group II: MK-4716 + PembrolizumabExperimental Treatment2 Interventions
Group III: MK-4716 + CetuximabExperimental Treatment2 Interventions

Find a Clinic Near You

Who Is Running the Clinical Trial?

Merck Sharp & Dohme LLC

Lead Sponsor

Trials
4,096
Recruited
5,232,000+
Chirfi Guindo profile image

Chirfi Guindo

Merck Sharp & Dohme LLC

Chief Marketing Officer since 2022

Degree in Engineering from Ecole Centrale de Paris, MBA from New York University Stern School of Business

Robert M. Davis profile image

Robert M. Davis

Merck Sharp & Dohme LLC

Chief Executive Officer since 2021

JD from Northwestern University Pritzker School of Law, MBA from Northwestern University Kellogg Graduate School of Management, Bachelor's in Finance from Miami University

Citations

A Clinical Study of MK-4716 in People With Certain Solid ...

Subset of arm MK-4716 Dose Escalation and subset of arm MK-4716 + Cetuximab: Has a confirmed diagnosis of locally advanced unresectable or metastatic solid ...

Chemotherapeutic Effectiveness of Combining Cetuximab for ...

Our results showed that cetuximab could significantly prolong PFS and OS in mCRC patients with wild type KRAS, but did not remarkably improve ...

EMD Serono Trials

MK-4716, Pembrolizumab, Keytruda, Cetuximab. Merck Sharp & Dohme LLC ... COMBINATION WITH CETUXIMAB, IN COLORECTAL CANCER PATIENTS WITH MINIMAL RESIDUAL DISEASE ( ...

Long-term Survival and Molecular Biomarker Evaluation of ...

At a median follow-up of 47.4 months, median overall survival (OS) and 2-year OS rate were 12.7 months and 32% in all evaluable patients (n=88) ...

NCT06589804 | Testing the Addition of Anti-Cancer Drug ...

Giving cetuximab and pembrolizumab together may be more effective at treating patients with recurrent and/or metastatic HNSCC than pembrolizumab alone. Detailed ...

A Clinical Study of MK-4716 in People With Certain Solid ...

Blood samples will be collected to estimate Cmax of MK-4716. At designated timepoints (up to approximately 58 days). Trough Plasma Concentration (Ctrough) of MK ...

A Study of MK-4700 Alone or With Pembrolizumab in ...

The goal of this study is to learn about the safety of different doses of MK-4700 and if people tolerate them. The study will also measure what happens in a ...

Construction and Evaluation of Tumor Immunotherapy and ...

By integrating biochemical indicators and related hemodynamic data, it constructs a risk early-warning system for organ damage in patients ...

Everything Comes with a Price: The Toxicity Profile of DNA ...

This review provides a comprehensive overview on the safety profile of DDR-targeting agents, including indications for their management in clinical practice.