242 Participants Needed

HQP1351 for Leukemia

Recruiting at 9 trial locations
KS
BG
Overseen ByBill Garrett
Age: 18+
Sex: Any
Trial Phase: Phase 1
Sponsor: Ascentage Pharma Group Inc.
Must be taking: Tyrosine kinase inhibitors
No Placebo GroupAll trial participants will receive the active study treatment (no placebo)

What You Need to Know Before You Apply

What is the purpose of this trial?

This trial tests a new treatment called HQP1351, a potential drug for certain types of leukemia. It aims to determine the best dose and understand the drug's movement through the body. The trial targets individuals with chronic myeloid leukemia (CML) or acute lymphoblastic leukemia (ALL) who have tried at least two other treatments without success. Those who have experienced resistance or side effects from previous treatments and continue to struggle with their condition may be suitable candidates. As a Phase 1 trial, this research focuses on understanding how the treatment works in people, offering participants the opportunity to be among the first to receive this new drug.

Do I have to stop taking my current medications for the trial?

The trial requires that you stop taking any tyrosine kinase inhibitors (TKIs) at least 7 days before starting the study drug, HQP1351. If you are taking other medications that might interact with HQP1351, you may also need to stop those, but the protocol does not specify all such medications.

Is there any evidence suggesting that HQP1351 is likely to be safe for humans?

Research shows that HQP1351, also known as Olverembatinib, is generally well-tolerated by patients. Studies have found it can help people with certain types of leukemia who haven't responded well to other treatments. Reports from earlier trials indicate that patients experienced few serious side effects. For instance, one study found that HQP1351 was safe for people with chronic myeloid leukemia that didn't respond to other treatments. Another study confirmed its safety when used with another drug for a specific type of acute lymphoblastic leukemia.

In summary, current evidence suggests that HQP1351 is safe for people, with manageable side effects. However, as this trial is still in the early stages, more research is needed to fully understand its safety.12345

Why do researchers think this study treatment might be promising for leukemia?

Unlike the standard leukemia treatments, which often involve chemotherapy or targeted therapies like tyrosine kinase inhibitors (TKIs), HQP1351 is a new type of TKI that targets specific mutations in cancer cells more precisely. Researchers are excited about HQP1351 because it can overcome resistance to current TKIs, a major hurdle in treating leukemia effectively. This precision could lead to better outcomes for patients who haven't had success with existing options. Plus, its potential for fewer side effects makes it a promising alternative for long-term treatment.

What evidence suggests that HQP1351 might be an effective treatment for leukemia?

Research has shown that HQP1351, also known as olverembatinib, may help treat certain types of leukemia. In studies with patients who have chronic myeloid leukemia and a specific mutation called T315I, HQP1351 worked well and was generally safe. One study found that after 36 months, 57.1% of patients did not experience disease progression, and 69.6% were still alive. These results suggest that HQP1351 could be a good option for patients who have not had success with other treatments. Participants in this trial will join various treatment cohorts to further evaluate the effectiveness and safety of HQP1351.26789

Who Is on the Research Team?

YZ

Yifan Zhai, MD, PhD

Principal Investigator

Ascentage Pharma Group Inc.

Are You a Good Fit for This Trial?

This trial is for people with chronic myelogenous leukemia (CML) or Philadelphia chromosome-positive acute lymphoblastic leukemia (Ph+ ALL), who have not responded well to at least two tyrosine kinase inhibitors (TKIs). Participants must be able to follow the study procedures and agree to use effective contraception. Those with certain health conditions, recent surgeries, active infections like HIV or hepatitis, poorly controlled diabetes, or a history of other cancers within the last year are excluded.

Inclusion Criteria

You have previously received a second-line TKI treatment, but it did not work for you.
You have chronic myeloid leukemia (CML) in any phase (chronic, accelerated or blast crisis) or Philadelphia chromosome-positive acute lymphoblastic leukemia (Ph+ ALL). You may or may not have a specific T315I mutation.
You are expected to live for at least 3 more months.
See 19 more

Exclusion Criteria

Previously treated with HQP1351
You have recently received other treatments that are not allowed in this study.
You are currently taking medication to suppress your immune system, except for a short course of steroids.
See 17 more

Timeline for a Trial Participant

Screening

Participants are screened for eligibility to participate in the trial

2-4 weeks

Treatment

Participants receive HQP1351 orally every other day in 28-day cycles, with dose-limiting toxicity observation during the first cycle

28 days per cycle

Dose Escalation and Expansion

Cohort D involves dose escalation and expansion with HQP1351 and blinatumomab in 42-day cycles

42 days per cycle

Follow-up

Participants are monitored for safety and effectiveness after treatment

4 weeks

What Are the Treatments Tested in This Trial?

Interventions

  • HQP1351
Trial Overview The trial is testing HQP1351, a new drug for patients resistant to standard treatments for CML and Ph+ ALL. It's an open-label study where everyone knows what treatment they're getting. The goal is to find out how much of the drug can be safely given (the recommended phase 2 dose) and understand how it affects the body by studying its pharmacokinetics.
How Is the Trial Designed?
4Treatment groups
Experimental Treatment
Group I: Cohort DExperimental Treatment2 Interventions
Group II: Cohort CExperimental Treatment1 Intervention
Group III: Cohort BExperimental Treatment1 Intervention
Group IV: Cohort AExperimental Treatment1 Intervention

Find a Clinic Near You

Who Is Running the Clinical Trial?

Ascentage Pharma Group Inc.

Lead Sponsor

Trials
54
Recruited
5,700+

Citations

Olverembatinib (HQP1351), a well-tolerated and effective ...Olverembatinib (HQP1351), a well-tolerated and effective tyrosine kinase inhibitor for patients with T315I-mutated chronic myeloid leukemia.
Updated Results of Pivotal Phase 2 Trials of Olverembatinib ...At 36 months, the PFS rate was 57.1% (95% CI: 33.3%-75.1%) and the OS rate was 69.6% (95% CI: 46.6%-84.2%) (Figure 3). Six pts withdrew because ...
Ascentage Pharma to Present Data from Multiple Studies of ...As of July 24, 2025, 39 (83.0%) patients received at least one efficacy evaluation; 36 (76.6%) at least two efficacy evaluations; and 34 (72.3%) ...
Updated efficacy results of olverembatinib (HQP1351) in ...After a median follow-up of 17.0 (4.1-57.5) months, the median progression-free survival (PFS) was 25.7 months (12.1-not reached [NR]). Among ...
Olverembatinib Demonstrates Efficacy and Safety in ...Olverembatinib demonstrated preliminary efficacy and was well tolerated in patients with heavily pretreated chronic-phase myeloid leukemia.
Olverembatinib (HQP1351) Overcomes Resistance ...Olverembatinib is a well-tolerated TKI with potential to overcome resistance. This update presents efficacy and safety data from a phase 1b ...
Study of HQP1351 in Subjects With Refractory CML and ...RP2D of HQP1351 will be determined based on the comprehensive analyses of the PK, safety, and efficacy data of the US patients treated with HQP1351, when ...
Safety and Efficacy of Olverembatinib (HQP1351) ...These preliminary data showed that olverembatinib in combination with lisaftoclax appears to be a safe and effective regimen in patients with R/R Ph+ ALL. This ...
Olverembatinib (HQP1351), a well-tolerated and effective ...Olverembatinib was well tolerated, with significant antileukemic activity in adults with TKI-resistant CML-CP and CML-AP, especially those with the T315I ...
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