[18F]FTP PET/CT Imaging for Cocaine Addiction

Age: 18 - 65
Sex: Any
Trial Phase: Phase 1 & 2
Sponsor: University of Pennsylvania
No Placebo GroupAll trial participants will receive the active study treatment (no placebo)

What You Need to Know Before You Apply

What is the purpose of this trial?

This trial explores a new method to understand how the brain's D3 dopamine receptors, which are involved in mood, thought, and addiction, function in individuals with cocaine addiction and healthy volunteers. It employs a special PET/CT scan with a compound called [18F]FTP, a radiotracer used in imaging, to obtain clearer images of these brain receptors. The trial includes different groups: one consists of healthy individuals who may receive either a placebo or a calming medicine called lorazepam before scanning, and another involves those seeking treatment for cocaine addiction. This trial suits males who have been using cocaine regularly and seek help with their addiction, as well as healthy volunteers without major health issues or certain mental health conditions. Participants must have a recent brain MRI or be willing to undergo one for the study. As a Phase 1, Phase 2 trial, this research aims to understand how the treatment works in people and measure its effectiveness in an initial, smaller group.

Will I have to stop taking my current medications?

The trial requires that participants do not use dopaminergic CNS stimulants (medications affecting the central nervous system) within 30 days of screening. Additionally, cocaine-dependent participants cannot be on any psychoactive medications. Other medications may be allowed if they do not interfere with the study, but it's best to discuss your specific medications with the study team.

What prior data suggests that this protocol is safe for imaging D3 receptors in the brain?

Research has shown that [18F]FTP, used in PET/CT scans, has been tested for safety in both animals and humans. In animal studies, researchers used [18F]FTP to track its movement through the body, and no harmful effects were found. In human studies, [18F]FTP is being evaluated for its ability to measure certain brain receptors related to conditions like addiction and some mental health issues.

Previous research using this imaging method has not identified any major safety problems, but ongoing testing aims to ensure its safety for people. As this trial is in the early stages, it primarily focuses on understanding how the treatment works in the body and ensuring participant safety.12345

Why are researchers excited about this trial?

Researchers are excited about the [18F]FTP PET/CT imaging trial for cocaine addiction because it explores a novel way to understand brain activity in cocaine-dependent individuals. Unlike traditional treatments that focus on managing withdrawal symptoms or reducing cravings through medication or therapy, this imaging approach aims to provide detailed insights into how cocaine affects the brain at a metabolic level. By using [18F]FTP, a radiotracer, alongside advanced PET/CT scans, researchers hope to map out specific brain changes in cocaine users, offering a clearer picture that could lead to more targeted and effective treatments in the future. This method not only helps in assessing current brain function but also in comparing these findings with healthy individuals, potentially revolutionizing how cocaine addiction is understood and treated.

What evidence suggests that [18F]FTP PET/CT is effective for imaging D3 receptors in cocaine addiction?

Studies have shown that PET imaging, part of the [18F]FTP PET/CT process, effectively detects brain changes related to cocaine addiction. This trial includes several cohorts using [18F]FTP PET/CT to study different aspects of cocaine addiction. For instance, Cohort 3 involves cocaine-dependent males undergoing imaging to determine arterial blood input and FTP parent to metabolite ratio curves. Meanwhile, Cohort 4 examines test/retest variability in cocaine-dependent patients. This imaging method identifies specific brain areas affected by cocaine use, which is crucial for understanding addiction. Research has also shown that brain imaging can monitor changes in brain activity when cocaine use stops. This makes [18F]FTP PET/CT a promising tool for understanding cocaine's impact on the brain and potentially guiding treatment options.23467

Who Is on the Research Team?

Jacob G. Dubroff, MD, PhD profile ...

Jacob Dubroff, MD, PhD

Principal Investigator

University of Pennsylvania

Are You a Good Fit for This Trial?

This trial is for healthy males aged 18-60, or those with moderate to severe cocaine use disorder seeking treatment. Participants must be in good health as determined by an investigator and not have significant medical conditions that could affect the study or their safety. Pregnant women, individuals with certain medical conditions like liver disease, epilepsy, or severe respiratory issues are excluded.

Inclusion Criteria

I am a male aged between 18 and 60 years and have a dependence on cocaine.
I primarily use cocaine by smoking it.
Participants for Cohort 1 and 2 (Healthy Volunteers) must be in good general health as determined by the investigator
See 4 more

Exclusion Criteria

I have not had a head injury that affects brain scans.
I am not pregnant.
Participants with current alcohol consumption exceeding 25 drinks per week are excluded
See 11 more

Timeline for a Trial Participant

Screening

Participants are screened for eligibility to participate in the trial

2-4 weeks

Imaging and Treatment

Participants undergo dynamic [18F]FTP PET/CT brain scans with different interventions (lorazepam, perphenazine, or placebo) and arterial sampling for cocaine-dependent subjects

2 days per participant
2 visits (in-person)

Test/Retest

Participants undergo test-retest scans to evaluate the variability of [18F]FTP uptake measures

2 days per participant
2 visits (in-person)

Follow-up

Participants are monitored for safety and effectiveness after imaging procedures

4 weeks

What Are the Treatments Tested in This Trial?

Interventions

  • [18F]FTP PET/CT
Trial Overview [18F]FTP PET/CT scans are being tested to measure D3 dopamine receptor binding in the brain. The study involves healthy volunteers and cocaine-dependent subjects who will receive either lorazepam or a placebo before scanning to assess [18F]FTP uptake variability.
How Is the Trial Designed?
4Treatment groups
Experimental Treatment
Group I: Cohort 4: Cocaine-dependent Test/RetestExperimental Treatment1 Intervention
Group II: Cohort 3: Arterial samplingExperimental Treatment1 Intervention
Group III: Cohort 2: Healthy Volunteer Test/RetestExperimental Treatment1 Intervention
Group IV: Cohort 1a: Lorazepam; 1b: PerphenazineExperimental Treatment1 Intervention

Find a Clinic Near You

Who Is Running the Clinical Trial?

University of Pennsylvania

Lead Sponsor

Trials
2,118
Recruited
45,270,000+

Published Research Related to This Trial

Neuroimaging has revealed that cocaine dependence affects not only dopamine-rich areas in the brain but also disrupts cortical regions, indicating a more complex network of brain dysfunction in addiction.
Recent studies suggest that changes in functional connectivity in cocaine users are linked to structural brain abnormalities, highlighting the potential for neuroimaging to inform personalized treatment strategies for addiction.
The use of brain imaging to elucidate neural circuit changes in cocaine addiction.Hanlon, CA., Canterberry, M.[2021]

Citations

Fluorodeoxyglucose-Positron Emission Tomography in Rats ...Biomarkers that are indicative of recreational drug use and addicted behavior are lacking. We performed a translational [18F]-fluorodeoxyglucose-positron ...
Brain Imaging Studies of the Effects of Cocaine Abstinence ...1. Cocaine abstinent group. Interventions: Radiation: PET scan; Other: fMRI · 2. Normal healthy control group. Interventions: Radiation: PET scan; Other: fMRI.
PET Imaging of the Effects of Age and Cocaine on the ...Here we report our preliminary studies evaluting the NET in individuals with cocaine dependence (COC) in comparison to healthy controls (HC) using (S,S)-[11C] ...
[18F]FTP PET/CT Imaging for Cocaine AddictionThe research highlights that PET imaging, which is part of the [18F]FTP PET/CT treatment, is effective in identifying brain changes associated with cocaine ...
A prospective 18F-fluorodeoxyglucose positron emission ...Conclusion: HIV infection and cocaine usage were independently associated with a decrease in brain glucose uptake as measured by 18F-FDG PET/CT.
Study Details | NCT02815917 | Evaluation of D3 Receptor ...Test-retest scans will evaluate the variability of [18F]FTP uptake measures in both healthy volunteer subjects and cocaine-dependent subjects. Official Title.
specific PET radioligand [18F]FluorTriopride estimated ...The objective of this study is to deter- mine the organ distribution of [18F]FTP in rodent and nonhuman primate species of animals to estimate ...
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