CVL-231 for Schizophrenia

No longer recruiting at 1 trial location
Age: 18 - 65
Sex: Any
Trial Phase: Phase 1
Sponsor: Cerevel Therapeutics, LLC
No Placebo GroupAll trial participants will receive the active study treatment (no placebo)

What You Need to Know Before You Apply

What is the purpose of this trial?

This trial tests an experimental treatment, CVL-231 (also known as Emraclidine), to observe its effects on certain brain receptors. The main focus is to understand how well this drug interacts with muscarinic receptors type 4 in the brain after oral administration. The trial seeks healthy men and women (who cannot have children) between 18 and 55 years old. Participants should not have any major health issues or a history of psychiatric disorders. As a Phase 1 trial, this research aims to understand how the treatment works in people, offering participants the opportunity to be among the first to receive this new treatment.

Do I need to stop my current medications to join the trial?

The trial information does not specify whether you need to stop taking your current medications. It's best to discuss this with the trial team or your doctor.

Is there any evidence suggesting that CVL-231 is likely to be safe for humans?

Research shows that CVL-231, also known as emraclidine, is under study for its safety in humans. These studies focus on adults with schizophrenia to assess its long-term safety and tolerability. The goal is to ensure the treatment does not cause serious side effects with ongoing use.

Although detailed results from these studies are not yet available, the testing of CVL-231 in humans suggests it demonstrated some safety in earlier tests, often conducted on animals or in a lab.

CVL-231 works by affecting certain parts of the brain, potentially reducing symptoms without causing major harm. However, like any new treatment, risks may exist. Joining a clinical trial involves understanding these risks. Consulting a healthcare provider can help determine if participating in a trial is appropriate.12345

Why do researchers think this study treatment might be promising?

Researchers are excited about CVL-231 because it offers a novel approach to treating conditions like schizophrenia. Unlike standard treatments that generally target dopamine receptors, CVL-231 focuses on muscarinic receptors in the brain, which may result in fewer side effects like weight gain or sedation. This unique mechanism of action could potentially provide a more effective and tolerable treatment option for patients.

What evidence suggests that CVL-231 might be an effective treatment for muscarinic receptor occupancy in the brain?

Research shows that CVL-231, the investigational treatment in this trial, may help treat schizophrenia. In earlier studies, patients taking CVL-231 experienced fewer core symptoms of schizophrenia. Importantly, most participants tolerated CVL-231 well in these studies. The drug affects certain brain receptors that help control mood and perception. Early results suggest this method could manage symptoms without many common side effects of other treatments. While more research is needed, these initial findings are promising.26789

Who Is on the Research Team?

ML

Matthew Leoni, MD, MBA

Principal Investigator

Cerevel Therapeutics, LLC

Are You a Good Fit for This Trial?

Inclusion Criteria

Capable of providing informed consent and following study requirements
Sexually active men with a pregnant or a nonpregnant partner of childbearing potential must agree to use a double-barrier method of birth control, including a condom, and practice contraception during treatment and through 7 days post dose

Exclusion Criteria

You have used any tobacco or nicotine products in the past month.
Subjects with a 12-lead ECG demonstrating either of the following (average of 3 ECGs obtained at the Screening Visit): QT interval corrected for heart rate using Fridericia's formula >450 msec, Left ventricular hypertrophy, Orthostatic hypotension, which is defined as a decrease of ≥20 mmHg in systolic blood pressure and/or a decrease of ≥10 mmHg in diastolic blood pressure after at least 3 minutes of standing compared with the immediately previous supine/semi-recumbent blood pressure at Screening or at the prescan time point prior to baseline PET scan.
Subjects with a current or past personal history of any psychiatric disorder as classified by DSM-5 criteria or immediate family members with any psychiatric disorder as classified by DSM-5 criteria that require treatment
See 9 more

Timeline for a Trial Participant

Screening

Participants are screened for eligibility to participate in the trial

1-2 weeks

Treatment

Participants receive a single oral dose of CVL-231 and undergo PET scans to evaluate M4 receptor occupancy

1 day
1 visit (in-person)

Follow-up

Participants are monitored for safety and effectiveness after treatment, including suicidality assessment

10 days
2 visits (in-person)

What Are the Treatments Tested in This Trial?

Interventions

  • CVL-231
How Is the Trial Designed?
1Treatment groups
Experimental Treatment
Group I: CVL-231Experimental Treatment1 Intervention

Find a Clinic Near You

Who Is Running the Clinical Trial?

Cerevel Therapeutics, LLC

Lead Sponsor

Trials
37
Recruited
5,500+

Citations

A Trial of 10 and 30 mg Doses of CVL-231 (Emraclidine) in ...This is a Phase 2, multicenter, randomized, double-blind, placebo-controlled, parallel-group, 6-week trial to evaluate the efficacy, safety, and tolerability ...
A Study to Evaluate Safety and Tolerability of CVL-231 ...The primary purpose of this study is to assess the long-term safety and tolerability of oral emraclidine in adult participants with schizophrenia.
AbbVie Provides Update on Phase 2 Results for ...AbbVie (NYSE: ABBV) today announced that its two Phase 2 EMPOWER trials investigating emraclidine as a once-daily, oral monotherapy treatment for adults with ...
A Trial of 15 and 30 mg Doses of CVL-231 (Emraclidine) in ...This is a Phase 2, multicenter, randomized, double-blind, placebo-controlled, parallel-group, 6-week trial to evaluate the efficacy, safety, ...
Emraclidine (CVL-231) to treat acute psychosis in ...Although these drugs are effective in reducing core symptoms of schizophrenia, undesirable adverse effects, such as tardive dyskinesia (a disorder causing ...
Material Safety Data Sheet of Emraclidine (CVL-231)Material Safety Data Sheet of Emraclidine (CVL-231) contains identification of substance and details of the supplier of the safety data sheet.
Emraclidine (CAS 2170722-84-4)Emraclidine. Item No. 42125. Emraclidine (CVL-231, PF-06852231, CAS Number: 2170722-84. Download Product Insert (PDF)Download Safety Data Sheet (SDS) (PDF). 5 ...
Emraclidine | CVL231 | PAM of M4 mAChR | Axon 4086Emraclidine is a brain-penetrant, highly selective M4 receptor positive allosteric modulator. More Information. Certificates. Certificate of Analysis (B1).
A Study to Evaluate Safety and Tolerability of CVL-231 ...The primary purpose of this study is to assess the long-term safety and tolerability of oral emraclidine in adult participants with schizophrenia.
Unbiased ResultsWe believe in providing patients with all the options.
Your Data Stays Your DataWe only share your information with the clinical trials you're trying to access.
Verified Trials OnlyAll of our trials are run by licensed doctors, researchers, and healthcare companies.
Terms of Service·Privacy Policy·Cookies·Security