Trametinib for Advanced Cancer

No longer recruiting at 11 trial locations
No Placebo GroupAll trial participants will receive the active study treatment (no placebo)
Breakthrough TherapyThis drug has been fast-tracked for approval by the FDA given its high promise
Approved in 4 JurisdictionsThis treatment is already approved in other countries

What You Need to Know Before You Apply

What is the purpose of this trial?

This trial tests the safety and effectiveness of trametinib for people with advanced cancer, particularly those whose cancer resists usual treatments. Trametinib blocks certain proteins that aid cancer cell growth, potentially stopping or killing the cancer. The trial focuses on individuals with liver problems that often hinder standard treatments. People with advanced cancer unresponsive to other treatments and who have liver issues might be suitable for this trial. As a Phase 1 trial, the research aims to understand how the treatment works in people, offering participants a chance to be among the first to receive this potentially groundbreaking therapy.

Do I have to stop taking my current medications for the trial?

The trial does not specify if you need to stop taking your current medications, but you cannot use other anti-cancer therapies or herbal supplements during the study. It's best to discuss your specific medications with the study team.

Is there any evidence suggesting that trametinib is likely to be safe for humans?

Research has shown that trametinib, a drug under study for advanced cancer, has safety information from past studies. In earlier research with melanoma patients, trametinib was tested and found to have some side effects. A small number of people experienced a serious fever, known as pyrexia, with about 5% requiring hospital care. Other side effects included rash and high blood pressure, which were serious but not very common.

The FDA has already approved trametinib for treating certain types of cancer when used with other drugs. This approval suggests that trametinib is generally considered safe enough for use, though monitoring for side effects remains important.

Overall, while trametinib carries some risks, it has been tested in humans before and shows promise for treating advanced cancers.12345

Why do researchers think this study treatment might be promising?

Trametinib is unique because it targets a specific pathway involved in cancer cell growth called the MEK pathway, which is different from many standard treatments that often focus on other parts of the cell cycle. This targeted approach can potentially lead to more precise attacks on cancer cells while sparing healthy ones, reducing side effects. Researchers are excited about trametinib because it offers a new way to tackle advanced cancers, especially for patients who may not respond well to traditional chemotherapy or radiation therapies.

What evidence suggests that trametinib might be an effective treatment for advanced cancer?

Research has shown that trametinib, the treatment under study in this trial, can slow the growth of certain cancers. In one study, patients taking trametinib lived an average of 4.9 months without their cancer worsening, compared to just 1.5 months for those not taking it. Additionally, after five years, many patients on trametinib lived longer. This suggests that trametinib, which blocks proteins necessary for cancer cell growth, may help manage advanced cancers, even in patients with liver problems where usual treatments might not work. While more research is needed, these findings offer promise for those considering participation in clinical trials with trametinib.678910

Who Is on the Research Team?

Dr. Lillian Siu - Ontario Institute for ...

Lillian Siu, MD

Principal Investigator

University Health Network Princess Margaret Cancer Center LAO

Are You a Good Fit for This Trial?

This trial is for patients with advanced cancers that can't be cured or controlled, including those with liver dysfunction. It includes people who've failed previous treatments like BRAF inhibitors for melanoma and have solid tumors such as pancreatic cancer. Participants must be able to take oral medication, have a life expectancy over 3 months, and not have had recent other treatments.

Inclusion Criteria

I can take pills and don't have major stomach or bowel issues affecting drug absorption.
Platelets >= 75 x 10^9/L
PT =< 1.5 x institutional ULN
See 33 more

Exclusion Criteria

I do not have any unmanaged ongoing illnesses.
I haven't taken any experimental drugs in the last 28 days.
I am not taking any medications that are not allowed in the study.
See 14 more

Timeline for a Trial Participant

Screening

Participants are screened for eligibility to participate in the trial

2-4 weeks

Treatment

Patients receive trametinib orally once daily on days 1-28. Cycles repeat every 28 days in the absence of disease progression or unacceptable toxicity.

28 days per cycle

Follow-up

Participants are monitored for safety and effectiveness after treatment

4 weeks

What Are the Treatments Tested in This Trial?

Interventions

  • Trametinib
Trial Overview The trial is testing Trametinib's effectiveness and safe dosage in advanced cancer patients with varying levels of liver function. The drug aims to block proteins essential for cancer cell growth which may stop the spread of the disease especially in those typically excluded from trials due to hepatic dysfunction.
How Is the Trial Designed?
1Treatment groups
Experimental Treatment
Group I: Treatment (trametinib)Experimental Treatment1 Intervention

Trametinib is already approved in European Union, United States, Canada, Japan for the following indications:

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Approved in European Union as Mekinist for:
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Approved in United States as Mekinist for:
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Approved in Canada as Mekinist for:
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Approved in Japan as Mekinist for:

Find a Clinic Near You

Who Is Running the Clinical Trial?

National Cancer Institute (NCI)

Lead Sponsor

Trials
14,080
Recruited
41,180,000+

Citations

Five-Year Outcomes with Dabrafenib plus Trametinib in ...The progression-free survival rates were 21% (95% confidence interval [CI], 17 to 24) at 4 years and 19% (95% CI, 15 to 22) at 5 years.
2.pubmed.ncbi.nlm.nih.govpubmed.ncbi.nlm.nih.gov/31166680/
Five-Year Outcomes with Dabrafenib plus Trametinib in ...The progression-free survival rates were 21% (95% confidence interval [CI], 17 to 24) at 4 years and 19% (95% CI, 15 to 22) at 5 years.
3.pubmed.ncbi.nlm.nih.govpubmed.ncbi.nlm.nih.gov/30690294/
Five-year outcomes from a phase 3 METRIC study in ...Five-year results of efficacy and safety analyses are reported. Results: The median PFS was 4.9 months in the trametinib arm versus 1.5 months in the ...
Real-world efficacy of the dabrafenib-trametinib (D-T) ...The findings confirmed the significant efficacy of DT in combination with BRAF V600E-mutated metastatic NSCLC in pretreated and untreated patients.
Results of the study GEM1801. | Journal of Clinical OncologyIn patients who had a complete response, the 5-year OS rate was 58.3% (95% CI: 31.3-100) while the median overall survival was not reached. In ...
Activity of the MEK Inhibitor Trametinib (GSK1120212) in ...We report the results of melanoma patients treated in the Phase I, first-in-human study of trametinib for patients with advanced malignancies. The main ...
Mekinist - accessdata.fda.govGrade 3-4 pyrexia occurred in 4.3% of patients, hospitalizations due to pyrexia occurred in 5.1% of patients, pyrexia with complications (dehydration, ...
Safety profile of TAFINLAR® (dabrafenib) + MEKINIST® ...TAFINLAR® (dabrafenib) and MEKINIST® (trametinib) safety profile in melanoma from clinical studies. For UK healthcare professionals only.
BRAF and MEK Inhibitors and Their Toxicities: A Meta-AnalysisThe most common AEs of grade 3 or higher were pyrexia, rash, and hypertension for Dabrafenib + Trametinib (6%), rash and hypertension for Encorafenib + ...
Updated efficacy and safety data of dabrafenib (D) ...Conclusions: D + T combination therapy continues to significantly improve outcomes in ATC, with a favorable safety profile. This regimen represents a clinically ...
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