LY3410738 for Solid Tumors

Not currently recruiting at 46 trial locations
PA
Overseen ByPatient Advocacy
No Placebo GroupAll trial participants will receive the active study treatment (no placebo)

What You Need to Know Before You Apply

What is the purpose of this trial?

This trial examines the safety and early effectiveness of a new treatment, LY3410738 (an experimental treatment), alone or combined with other drugs, for individuals with advanced solid tumors that have specific genetic changes (mutations in IDH1 or IDH2 genes). It includes conditions such as cholangiocarcinoma, chondrosarcoma, and glioma. Participants must have a confirmed IDH mutation and an advanced solid tumor that does not respond to standard treatments. This trial may suit those with these specific tumor types that no longer respond to other treatments. As a Phase 1 trial, the research focuses on understanding how the treatment works in people, offering participants the opportunity to be among the first to receive this new treatment.

Do I need to stop my current medications to join the trial?

The trial protocol does not clearly specify if you need to stop taking your current medications. However, you cannot participate if you are currently on certain strong CYP3A4 inhibitors or inducers, or P-gp inhibitors. It's best to discuss your specific medications with the trial team.

Is there any evidence suggesting that this trial's treatments are likely to be safe?

Research has shown that LY3410738 has been tested in several studies for safety in people with certain advanced solid tumors. Previous patients generally tolerated the treatment well.

In these studies, some patients experienced side effects. The most common were fatigue, nausea, and low blood counts, which can make it harder for the body to fight infections. However, these side effects were usually mild or manageable.

As this is a Phase 1 trial, the main goal is to assess the safety of LY3410738 and determine the best dose. The treatment is still being tested to ensure its safety for humans.

Prospective participants should discuss any concerns with their doctor and understand the potential risks and benefits before joining this trial.12345

Why are researchers excited about this trial's treatments?

Researchers are excited about LY3410738 because it offers a novel approach to treating solid tumors. Unlike traditional chemotherapy drugs, LY3410738 is designed to target specific mutations in cancer cells, potentially leading to more effective and less toxic treatments. Additionally, in combination with gemcitabine and cisplatin or durvalumab, LY3410738 may enhance the overall treatment effectiveness by leveraging multiple mechanisms of action. This targeted approach could provide a significant advance over standard therapies, which often involve broader-acting treatments that can harm healthy cells along with cancerous ones.

What evidence suggests that LY3410738 could be an effective treatment for advanced solid tumors?

Research shows that LY3410738 may help treat tumors with specific genetic changes. Earlier studies found that it slowed tumor growth in certain types of bile duct cancer and brain tumors with these genetic changes. In this trial, participants may receive LY3410738 alone or with chemotherapy drugs like gemcitabine and cisplatin, which previously showed a success rate of 42.1%. Early trials also demonstrated that LY3410738 alone reduced tumor growth by more than 60% in lab tests. These results suggest that LY3410738 could be a promising treatment for patients with these specific genetic mutations in their tumors.23467

Who Is on the Research Team?

C1

Call 1-877-CTLILLY (1-877-285-4559) or 1-317-615-4559 Mon - Fri 9 AM - 5 PM Eastern time (UTC/GMT - 5 hours, EST)

Principal Investigator

Eli Lilly and Company

Are You a Good Fit for This Trial?

Adults with advanced solid tumors that have specific mutations (IDH1 R132, IDH2 R140, or IDH2 R172) and are not responding to standard treatments. They should be in good physical condition (ECOG 0-1), able to swallow pills, and willing to use birth control. People who've had certain prior treatments or have active infections, uncontrolled diseases, brain metastases requiring steroids, or a history of severe immune-related side effects from other drugs can't join.

Inclusion Criteria

Measurable disease as determined by RECIST 1.1.
History of hypersensitivity to durvalumab or any excipient.
My cholangiocarcinoma has specific IDH1 or IDH2 mutations.
See 28 more

Exclusion Criteria

I haven't taken any cancer drugs or investigational treatments in the last 2 to 4 weeks.
I have cholangiocarcinoma and have not undergone specific liver treatments in the last 4 weeks, nor do I have complications like ascites, encephalopathy, ongoing cholangitis, mixed cancer types, or a liver transplant history.
I have not had major surgery in the last 4 weeks.
See 14 more

Timeline for a Trial Participant

Screening

Participants are screened for eligibility to participate in the trial

2-4 weeks

Dose Escalation

Phase 1 dose escalation to determine the maximum tolerated dose of LY3410738

8-12 weeks

Dose Expansion

Phase 1 dose expansion to further evaluate safety and clinical activity in multiple cohorts

16-24 weeks

Follow-up

Participants are monitored for safety and effectiveness after treatment

4 weeks

What Are the Treatments Tested in This Trial?

Interventions

  • LY3410738
Trial Overview The trial is testing LY3410738—an oral drug—on its own for safety and early signs of effectiveness against tumors with particular genetic changes. It's an open-label study where everyone knows what treatment they're getting. The trial includes patients with cancers like cholangiocarcinoma and glioma after some previous treatments failed.
How Is the Trial Designed?
2Treatment groups
Experimental Treatment
Group I: LY3410738 alone or in combination with gemcitabine and cisplatin or in combination with durvalumabExperimental Treatment4 Interventions
Group II: LY3410738Experimental Treatment1 Intervention

Find a Clinic Near You

Who Is Running the Clinical Trial?

Eli Lilly and Company

Lead Sponsor

Trials
2,708
Recruited
3,720,000+
Dr. Daniel Skovronsky profile image

Dr. Daniel Skovronsky

Eli Lilly and Company

Chief Medical Officer since 2018

MD from Harvard Medical School

David A. Ricks profile image

David A. Ricks

Eli Lilly and Company

Chief Executive Officer since 2017

BSc from Purdue University, MBA from Indiana University

Loxo Oncology, Inc.

Industry Sponsor

Trials
72
Recruited
11,600+

Jacob Van Naarden

Loxo Oncology, Inc.

Chief Executive Officer since 2019

A.B. in Molecular Biology from Princeton University

Dr. Jennifer Low

Loxo Oncology, Inc.

Chief Medical Officer since 2014

MD and PhD from Georgetown University; Undergraduate degree from California Institute of Technology

Citations

Final Results from a First-in-Human Phase I Study of the Dual ...LY3410738 plus CISGEM demonstrated a response rate of 42.1%, a median duration of response of 8.1 months, and a median progression-free survival ...
2.pubmed.ncbi.nlm.nih.govpubmed.ncbi.nlm.nih.gov/41026608/
Final Results from a First-in-Human Phase 1 Study of the ...Conclusions: LY3410738 demonstrated largely cytostatic antitumor activity in IDH1- or IDH2-mutated cholangiocarcinoma and IDH1-mutated gliomas.
NCT04521686 | Study of LY3410738 Administered to ...This is an open-label, multicenter Phase 1 study to evaluate safety, tolerability and preliminary efficacy of oral LY3410738 in patients with IDH1 R132-mutant ...
SO-1 A first-in-human phase 1 study of LY3410738 ...In an IDH1m CCA PDX model, single agent LY3410738 (10-30 mpk, QD) demonstrated >60% tumor growth inhibition. In a combination PDX study, LY3410738 (30 mpk, QD) ...
A phase I study of LY3410738, a first-in-class covalent ...This is an open-label, multicenter, global phase 1 study with oral LY3410738 currently enrolling patients with advanced CCA and other solid tumor types.
NCT04521686 | Study of LY3410738 Administered to ...This is an open-label, multicenter Phase 1 study to evaluate safety, tolerability and preliminary efficacy of oral LY3410738 in patients with IDH1 R132-mutant ...
Clinical TrialsThis is an open-label, multicenter Phase 1 study to evaluate safety, tolerability and preliminary efficacy of oral LY3410738 in patients with ...
Unbiased ResultsWe believe in providing patients with all the options.
Your Data Stays Your DataWe only share your information with the clinical trials you're trying to access.
Verified Trials OnlyAll of our trials are run by licensed doctors, researchers, and healthcare companies.
Terms of Service·Privacy Policy·Cookies·Security