Cimetidine for Protoporphyria

No longer recruiting at 2 trial locations
AK
PY
Overseen ByPaul Y Jiang
Prior Safety DataThis treatment has passed at least one previous human trial
Approved in 4 JurisdictionsThis treatment is already approved in other countries

What You Need to Know Before You Apply

What is the purpose of this trial?

This trial tests whether cimetidine (also known as Tagamet) can help individuals with erythropoietic protoporphyria (EPP) or X-linked protoporphyria (XLP). These conditions cause painful skin reactions to sunlight. The trial aims to determine if cimetidine can reduce these reactions and improve quality of life. Participants must have a history of painful skin reactions to light without blistering and must have participated in a previous study related to these conditions. As a Phase 2 trial, the research focuses on measuring the treatment's effectiveness in an initial, smaller group of people.

Will I have to stop taking my current medications?

The trial protocol does not specify if you must stop taking your current medications, but it mentions that any drugs or supplements that might interfere with safety or study objectives could be restricted. It's best to discuss your current medications with the study team.

Is there any evidence suggesting that cimetidine is likely to be safe for humans?

Research has shown that cimetidine is safe for people with porphyria, a group of disorders affecting the skin and nervous system. Studies and patient feedback suggest it is generally safe. However, concerns exist about long-term use. Safety information indicates that prolonged or repeated use might harm organs like the liver, kidneys, and testis. Most reports indicate that during cimetidine treatment, patients experienced reduced skin sensitivity to light, which benefits those with protoporphyria. Overall, while cimetidine is mostly well-tolerated, monitoring during treatment is important to ensure safety.12345

Why do researchers think this study treatment might be promising?

Researchers are excited about using Cimetidine for protoporphyria because it offers a unique approach compared to existing treatments. Most current therapies focus on managing symptoms or minimizing triggers, but Cimetidine, an H2-receptor antagonist commonly used to reduce stomach acid, may help by altering the metabolism of porphyrins, the compounds that accumulate in this condition. This novel mechanism could provide a new way to reduce the severity of symptoms in patients with protoporphyria, potentially improving quality of life where other treatments fall short.

What evidence suggests that cimetidine might be an effective treatment for protoporphyria?

Research has shown that cimetidine, which participants in this trial may receive, helps reduce symptoms in patients with other types of porphyria, such as acute intermittent porphyria. One study found that 15 out of 18 patients with erythropoietic protoporphyria who took cimetidine for at least four months experienced a noticeable decrease in symptoms. Cimetidine slows down the production of heme, which can help manage symptoms related to light sensitivity in protoporphyria. While more research is needed specifically for erythropoietic and X-linked protoporphyria, early results suggest it may be beneficial.46789

Who Is on the Research Team?

AK

Amy K Dickey, MD

Principal Investigator

Massachusetts General Hospital

KA

Karl E Anderson, MD

Principal Investigator

University of Texas

Are You a Good Fit for This Trial?

This trial is for individuals at least 15 years old with a confirmed diagnosis of Erythropoietic Protoporphyria (EPP) or X-linked Protoporphyria (XLP), who have a history of skin sensitivity to light but are not using other experimental therapies. Participants must be willing to use their smartphone for the study and expose themselves to light weekly.

Inclusion Criteria

I am 15 years old or older.
I am diagnosed with EPP or XLP and enrolled in the PC Study 7201.
I am willing and able to follow the study's procedures and give informed consent.
See 1 more

Exclusion Criteria

I have high porphyrin levels due to liver or bone marrow disease.
You have a known or suspected allergy or intolerance to cimetidine.
I have moderate to severe problems with my kidneys.
See 8 more

Timeline for a Trial Participant

Screening

Participants are screened for eligibility to participate in the trial

2-4 weeks

Treatment Period 1

Participants receive either placebo or cimetidine for 3 months

3 months
Visits before and after treatment period

Wash-out

A 3-month wash-out period to eliminate carry-over effects

3 months

Treatment Period 2

Participants receive the alternate treatment (cimetidine or placebo) for 3 months

3 months
Visits before and after treatment period

Follow-up

Participants are monitored for safety and effectiveness after treatment

4 weeks

What Are the Treatments Tested in This Trial?

Interventions

  • Cimetidine
  • Placebo
Trial Overview The trial is testing if oral Cimetidine can treat protoporphyrias by reducing protoporphyrin levels, improving tolerance to light, and enhancing quality of life. It's compared against a placebo, with outcomes measured through questionnaires and blood tests.
How Is the Trial Designed?
2Treatment groups
Active Control
Placebo Group
Group I: CimetidineActive Control1 Intervention
Group II: PlaceboPlacebo Group1 Intervention

Cimetidine is already approved in European Union, United States, Canada, Japan for the following indications:

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Approved in European Union as Tagamet for:
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Approved in United States as Tagamet for:
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Approved in Canada as Tagamet for:
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Approved in Japan as Tagamet for:

Find a Clinic Near You

Who Is Running the Clinical Trial?

Amy K. Dickey, M.D.

Lead Sponsor

Trials
1
Recruited
20+

The University of Texas Medical Branch, Galveston

Collaborator

Trials
263
Recruited
55,400+

University of Texas

Collaborator

Trials
193
Recruited
143,000+

Wake Forest University Health Sciences

Collaborator

Trials
1,432
Recruited
2,506,000+

Citations

1.pubmed.ncbi.nlm.nih.govpubmed.ncbi.nlm.nih.gov/27410690/
Novel Treatment Using Cimetidine for Erythropoietic ...Cimetidine has been shown to inhibit heme biosynthesis and results in symptomatic improvement in patients with acute intermittent porphyria (AIP) ...
Cimetidine for erythropoietic protoporphyriaThis study reports 18 cases treated with cimetidine at our department. Of them 15 completed at least 4 months of treatment resulting in a significant reduction ...
Effect of Oral Cimetidine in the ProtoporphyriasThe objective of this study is to determine the efficacy and safety of oral cimetidine administration for treatment of the protoporphyrias.
Cimetidine - StatPearls - NCBI Bookshelf - NIH... results in symptomatic improvement in children with acute intermittent porphyria and porphyria ... evidence for the benefit of cimetidine in protoporphyria.[8][9].
Effect of Oral Cimetidine in the ProtoporphyriasThe objective of this study is to determine the efficacy and safety of oral cimetidine administration for treatment of the protoporphyrias.
Cimetidine Formulation | Safety Data SheetH373 May cause damage to organs (Liver, Kidney, Testis) through prolonged or repeated exposure if swallowed. Precautionary Statements. : Prevention: P201 Obtain ...
Cimetidine Formulation | Safety Data SheetH373 May cause damage to organs (Liver, Kidney, Testis) through prolonged or repeated exposure if swallowed. Precautionary Statements. : Prevention: P201 Obtain ...
About Porphyria: Drug database... porphyria/: Safe in patients PV Tishler MD clinical data & patient reports: Safe ... Cimetidine, Tagamet, OK! www.drugs-porphyria.org: Not ...
Safety Data SheetRTECS Number. 51481-61-9 Cimetidine MF0035500. · Information on toxicological effects. · Acute toxicity: · LD/LC50 values that are relevant for ...
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