Hepcidin Mimetic for Polycythemia Vera

No longer recruiting at 16 trial locations
SD
Overseen ByStudy Director
Age: 18+
Sex: Any
Trial Phase: Phase 2
Sponsor: Protagonist Therapeutics, Inc.
Must be taking: Cytoreductive therapy
No Placebo GroupAll trial participants will receive the active study treatment (no placebo)
Prior Safety DataThis treatment has passed at least one previous human trial

What You Need to Know Before You Apply

What is the purpose of this trial?

This trial tests a treatment called PTG-300 (a hepcidin mimetic) for individuals with polycythemia vera, a condition where the body produces too many red blood cells, leading to frequent phlebotomies (blood removal procedures). The study aims to determine if PTG-300 is safe and effective in reducing the need for these phlebotomies. Participants will initially receive different doses of PTG-300, then either continue with PTG-300 or switch to a placebo, and finally return to PTG-300. This trial may suit adults diagnosed with polycythemia vera who require regular phlebotomies and are either not on cytoreductive therapy or are on a stable dose. As a Phase 2 trial, this research focuses on measuring the treatment's effectiveness in an initial, smaller group of people.

Will I have to stop taking my current medications?

If you are on cytoreductive therapy with hydroxyurea, interferon, or ruxolitinib, you can continue as long as your dose is stable or decreasing for at least 8 weeks before starting the trial. If you are not on these therapies, you must have stopped any prior cytoreductive therapy at least 24 weeks before joining the trial.

Is there any evidence suggesting that PTG-300 is likely to be safe for humans?

Research has shown that PTG-300, also known as rusfertide, has been tested in other studies to assess its safety in humans. In one study, patients with polycythemia vera, a blood disorder, experienced mostly mild side effects from rusfertide that did not cause major issues.

Another study found that rusfertide reduced the need for phlebotomy, a procedure to remove blood, and helped manage red blood cell levels without causing serious side effects.

While these results are encouraging, it is important to note that this trial remains in the middle stages of testing. More information is needed about its safety in larger groups. However, the results so far suggest that rusfertide is generally well-tolerated in people with polycythemia vera.12345

Why do researchers think this study treatment might be promising for polycythemia vera?

Unlike the standard treatments for polycythemia vera, such as phlebotomy, hydroxyurea, and interferon, PTG-300 offers a novel approach by mimicking the hormone hepcidin. Hepcidin plays a key role in regulating iron levels, which can help control red blood cell production without the need for frequent blood removal or cytotoxic agents. Researchers are excited because PTG-300 could offer a more targeted and potentially safer way to manage the condition, minimizing side effects and improving patients' quality of life. Additionally, the open-label extension in the trial suggests a commitment to understanding long-term benefits and safety of PTG-300.

What evidence suggests that PTG-300 might be an effective treatment for polycythemia vera?

Research has shown that PTG-300, also known as rusfertide, may help treat polycythemia vera, a condition where the body produces too many red blood cells. One study found that rusfertide helped maintain red blood cell levels below 45%, reducing the need for phlebotomies, which manage the condition. In this trial, participants will receive either PTG-300 or a placebo at different stages. Another study demonstrated that rusfertide was more effective than a placebo in controlling red blood cell levels. These findings suggest that PTG-300 could effectively manage polycythemia vera and reduce the need for frequent treatments.12678

Are You a Good Fit for This Trial?

Adults diagnosed with polycythemia vera, who've had regular phlebotomies for at least 28 weeks and are either on a stable or decreasing dose of cytoreductive therapy (like hydroxyurea, interferon, or ruxolitinib) for over 24 weeks. Those not on such therapies must have stopped them for at least 24 weeks prior.

Inclusion Criteria

You must meet ALL of the following inclusion criteria to be enrolled.
Records of all phlebotomies performed for at least 28 weeks (preferably up to 52 weeks) before dosing are available.
I've been on a stable or decreasing dose of specific blood cancer treatments for at least 8 weeks.
See 11 more

Exclusion Criteria

I have not had any active or chronic bleeding in the last 4 weeks.
I haven't had surgery under general anesthesia in the last month and don't plan any during the study.
I have been diagnosed with myelofibrosis following polycythemia vera.
See 1 more

Timeline for a Trial Participant

Screening

Participants are screened for eligibility to participate in the trial

2-4 weeks

Dose Finding

28 week dose finding phase to identify a dose that maintains hematocrit <45%

28 weeks

Randomized Withdrawal

12 week randomized withdrawal phase to confirm the response

12 weeks

Open-label Extension

Participants enter an up to 3 year open label extension to investigate long term safety

Up to 3 years

Follow-up

Participants are monitored for safety and effectiveness after treatment

4 weeks

What Are the Treatments Tested in This Trial?

Interventions

  • PTG-300
Trial Overview The trial is testing PTG-300, a hepcidin mimetic against a placebo in patients requiring frequent blood withdrawals due to polycythemia vera. It includes an initial phase where everyone gets PTG-300 to find the best dose followed by a blind test where neither doctors nor patients know who's getting what.
How Is the Trial Designed?
2Treatment groups
Experimental Treatment
Group I: Dose finding PTG-300 (Part 1); Placebo (Part 2); Open label extension PTG-300 (Part 3)Experimental Treatment2 Interventions
Group II: Dose finding PTG-300 (Part 1); PTG-300 (Part 2); Open label extension PTG-300 (Part 3)Experimental Treatment1 Intervention

Find a Clinic Near You

Who Is Running the Clinical Trial?

Protagonist Therapeutics, Inc.

Lead Sponsor

Trials
13
Recruited
960+

Citations

Results from VERIFY, a phase 3, double-blind, placebo ...Conclusions: In pts with PV receiving SOC, rusfertide resulted in a statistically significant reduction in the mean number of PHLs and improved ...
Final Results from the Phase 2 Revive Study Investigating the ...Preliminary results from the phase 2 REVIVE study (NCT04057040) demonstrated that rusfertide was superior to placebo in achieving hematocrit ( ...
Rusfertide, a Hepcidin Mimetic, for Control of Erythrocytosis ...In patients with polycythemia vera, rusfertide treatment was associated with a mean hematocrit of less than 45% during the 28-week dose-finding ...
Hepcidin Mimetics in Polycythemia Vera: Resolving the Irony ...Phase 2 trials demonstrate that rusfertide, a hepcidin mimetic, is highly effective in achieving and maintaining hematocrit below 45%, eliminating the need for ...
Rusfertide Demonstrates Promising Results in Phase 3 ...Protagonist and Takeda announce positive topline results from Phase 3 VERIFY study of rusfertide in patients with polycythemia vera.
Adding the Hepcidin Mimetic Rusfertide to the Standard of ...Rusfertide significantly improved multiple endpoints: reducing the need for phlebotomy, improving hematocrit control, and reducing symptoms ...
Study Details | NCT04057040 | Hepcidin Mimetic in ...The study is designed to monitor the PTG-300 safety profile and to obtain preliminary evidence of efficacy of PTG-300 for the treatment of phlebotomy-requiring ...
8.pubmed.ncbi.nlm.nih.govpubmed.ncbi.nlm.nih.gov/38381675/
Rusfertide, a Hepcidin Mimetic, for Control of Erythrocytosis ...Conclusions: In patients with polycythemia vera, rusfertide treatment was associated with a mean hematocrit of less than 45% during the 28-week ...
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