58 Participants Needed

Brexpiprazole for Bipolar Disorder

GB
PL
NK
Overseen ByNada Khalil, BA
Age: 18+
Sex: Any
Trial Phase: Phase 3
Sponsor: Douglas Mental Health University Institute
Must be taking: Mood stabilizers
Stay on Your Current MedsYou can continue your current medications while participating
No Placebo GroupAll trial participants will receive the active study treatment (no placebo)
Pivotal Trial (Near Approval)This treatment is in the last trial phase before FDA approval
Prior Safety DataThis treatment has passed at least one previous human trial
Approved in 6 JurisdictionsThis treatment is already approved in other countries

Trial Summary

What is the purpose of this trial?

Bipolar disorder (BD) is a frequent and lifelong recurrent mood disorder with treatment-resistant depressive episodes. Importantly, depressive symptoms and cognitive decline are major determinants of functionality and quality of life in this clinical population. There is robust evidence that individuals with BD have neurocognitive deficits (especially in memory and executive functioning domains) compared to the healthy population. These deficits are present in all mood states and can greatly affect patients' functional capacity, often more so than mood symptoms themselves. Many pharmacological treatments for BD adversely affect cognition, and those that are beneficial can be difficult to use. There is thus a pressing need to identify a safe, easy-to-use medication that can target both cognitive deficits and depressive symptoms in BD. It is expected that Brexpiprazole adjunctive treatment will be efficacious in treating BD type I and type II depression by improving mood symptoms, as well as cognitive capacity and global functioning, and that such changes will be accompanied by concurrent alterations in associated brain structures.

Do I have to stop taking my current medications for the trial?

The trial requires that you stop taking certain medications. You cannot participate if you are treated with fluoxetine, carbamazepine, risperidone, olanzapine, quetiapine (over 100mg/day), ziprazidone, or any other antipsychotic. However, you must be on a mood stabilizer like lithium, valproate, lamotrigine, or quetiapine (up to 100mg/day).

What data supports the idea that the drug Brexpiprazole for Bipolar Disorder is an effective treatment?

The available research shows that Brexpiprazole is effective for treating schizophrenia and as an additional treatment for major depressive disorder. It has been shown to improve symptoms and is generally well tolerated. However, there is no specific data provided about its effectiveness for treating Bipolar Disorder.12345

What safety data is available for Brexpiprazole?

Brexpiprazole, also known as Rexulti, is generally well tolerated with a relatively low incidence of activating and sedating adverse effects. It has been associated with moderate weight gain and small changes in metabolic parameters, which are not clinically significant. The most common adverse event is increased weight, with about 10% of patients gaining ≥7% body weight in short-term studies. Akathisia rates are low, and there are minimal effects on prolactin and the ECG QTc interval. Brexpiprazole is approved for schizophrenia and as an adjunct for major depressive disorder, with ongoing trials for other conditions.12346

Is the drug Brexpiprazole a promising treatment for Bipolar Disorder?

Brexpiprazole is a promising drug because it has been effective in treating major depressive disorder and schizophrenia, showing improvements in symptoms and being well tolerated by patients. It offers a new option for those who haven't fully responded to other treatments.12345

Research Team

SB

Serge Beaulieu, MD

Principal Investigator

Douglas Mental Health University Institute

Eligibility Criteria

Adults aged 18-75 with Bipolar I Disorder currently experiencing treatment-resistant depression, who have tried at least one other treatment without success. Participants must be on a mood stabilizer and have normal heart function. They cannot join if they are at high suicide risk, have psychotic symptoms, certain neurocognitive disorders, uncontrolled seizures, known allergies to Brexpiprazole or its components including lactose intolerance.

Inclusion Criteria

I have been diagnosed with Bipolar Disorder type I or II.
The following laboratory values are within normal limits at Screening: CBC with differential; ferritin; extended electrolytes (sodium, potassium, chloride, calcium, magnesium, phosphate); thyroid function test(s); kidney function tests; hemoglobin A1c; lipid profile; prolactin
I am taking a mood stabilizer like lithium, valproate, lamotrigine, or low-dose quetiapine.
See 1 more

Exclusion Criteria

I am not pregnant, breastfeeding, and I use birth control.
Drug abuse or dependence as per DSM-V (MINI)
I am lactose intolerant or have a similar condition.
See 20 more

Treatment Details

Interventions

  • Brexpiprazole
Trial OverviewThe trial is testing the effectiveness of Brexpiprazole as an additional treatment for depressive episodes in Bipolar I Disorder. It aims to improve mood symptoms and cognitive functions while monitoring changes in brain structures associated with these improvements.
Participant Groups
1Treatment groups
Experimental Treatment
Group I: PatientExperimental Treatment1 Intervention
Individuals diagnosed with Bipolar Disorder Type I or Type II and suffering a major depressive episode who will receive an adjunctive and variable dose of Brexpiprazole treatment

Find a Clinic Near You

Who Is Running the Clinical Trial?

Douglas Mental Health University Institute

Lead Sponsor

Trials
31
Recruited
2,800+

McMaster University

Collaborator

Trials
936
Recruited
2,630,000+

Jewish General Hospital

Collaborator

Trials
144
Recruited
283,000+

Findings from Research

Brexpiprazole is an effective new treatment for schizophrenia when used alone, providing a novel option for patients managing this condition.
Additionally, brexpiprazole can be used as an adjunctive therapy for major depressive disorder, enhancing the effectiveness of other treatments for individuals with this mental health issue.
Brexpiprazole (Rexulti): A New Monotherapy for Schizophrenia and Adjunctive Therapy for Major Depressive Disorder.Eaves, S., Rey, JA.[2022]
Brexpiprazole is an atypical antipsychotic that acts as a serotonin-dopamine activity modulator, showing efficacy as an adjunctive treatment for major depressive disorder (MDD) and schizophrenia, with its first approval in the USA in July 2015.
The drug functions by partially activating serotonin 1A and dopamine D2 receptors while blocking 5-HT2A and noradrenergic receptors, which may contribute to its therapeutic effects in various psychiatric disorders.
Brexpiprazole: First Global Approval.Greig, SL.[2018]
Brexpiprazole, a serotonin-dopamine activity modulator, has been shown to be more effective than standard antidepressant therapy alone in improving depressive symptoms in adults with major depressive disorder who did not fully respond to previous treatments, based on two phase III trials.
The drug was generally well tolerated over treatment periods of up to 52 weeks, suggesting a lower risk of activation-like side effects compared to similar medications like aripiprazole, making it a suitable adjunctive option for patients with persistent symptoms.
Adjunctive Brexpiprazole: A Review in Major Depressive Disorder.McKeage, K.[2018]

References

Brexpiprazole (Rexulti): A New Monotherapy for Schizophrenia and Adjunctive Therapy for Major Depressive Disorder. [2022]
Brexpiprazole: First Global Approval. [2018]
Adjunctive Brexpiprazole: A Review in Major Depressive Disorder. [2018]
Brexpiprazole: A Review in Schizophrenia. [2020]
Brexpiprazole: A Review in Schizophrenia. [2018]
Brexpiprazole for the Treatment of Schizophrenia: A Review of this Novel Serotonin-Dopamine Activity Modulator. [2016]