Upamostat for COVID-19 Prophylaxis

(PROTECT-APT 1 Trial)

No longer recruiting at 8 trial locations
ST
MF
ZH
Overseen ByZen Hafy, MD
Age: 18+
Sex: Any
Trial Phase: Phase 2
Sponsor: Henry M. Jackson Foundation for the Advancement of Military Medicine
Prior Safety DataThis treatment has passed at least one previous human trial

What You Need to Know Before You Apply

What is the purpose of this trial?

This trial aims to test the effectiveness and safety of a new treatment called Upamostat for people with COVID-19 or those exposed to the virus. The treatment is designed to prevent COVID-19 in individuals who have been in close contact with someone infected or to treat those who have recently tested positive and are showing symptoms. Suitable participants include adults who have tested positive for COVID-19 within the last five days and have at least two moderate symptoms, such as a sore throat or headache, or adults who were in close contact with someone with COVID-19 and have not yet developed symptoms. As a Phase 2 trial, the research focuses on measuring how well the treatment works in an initial, smaller group of people.

Will I have to stop taking my current medications?

The trial does not specify if you need to stop taking your current medications, but you cannot participate if you are taking or plan to start taking warfarin, apixaban (Eliquis), or rivaroxaban (Xarelto).

Is there any evidence suggesting that Upamostat is likely to be safe for humans?

Research shows that upamostat, the treatment under study, has been generally well-tolerated in past studies. One study found that it helped COVID-19 patients recover faster. Importantly, participants in that study did not experience severe side effects. This suggests that upamostat may be safe for people, but ongoing research will provide more information.12345

Why do researchers think this study treatment might be promising?

Unlike the standard of care for COVID-19, which often involves antiviral drugs like Remdesivir or monoclonal antibodies targeting the virus, Upamostat is unique because it works by inhibiting proteases crucial for the virus to replicate. This new mechanism of action means that Upamostat potentially stops the virus from spreading within the body at an earlier stage. Researchers are excited about Upamostat because it is an oral capsule, making it easier to administer and potentially more accessible than intravenous treatments. Additionally, its use as a prophylactic suggests it could prevent the onset of the disease, providing a proactive approach to managing COVID-19.

What evidence suggests that Upamostat might be an effective treatment for COVID-19?

In this trial, participants will receive either Upamostat or a placebo. Research has shown that Upamostat may help treat COVID-19. One study found that patients taking Upamostat had no hospitalizations, while those who did not take it did. Another study found that people recovered from severe COVID-19 symptoms in just 3 days on average. Upamostat works by blocking an enzyme that helps the virus spread in the body. These findings suggest that Upamostat could effectively manage COVID-19 symptoms and reduce the severity of the illness.34678

Who Is on the Research Team?

DC

Danielle Clark, PhD

Principal Investigator

Henry M. Jackson Foundation for the Advancement of Military Medicine

KP

Kristen Pettrone, MD

Principal Investigator

Henry M. Jackson Foundation for the Advancement of Military Medicine

Are You a Good Fit for This Trial?

This trial is for adults over 18 who've been in close contact with someone with confirmed COVID-19 or have mild symptoms within 5 days of onset. They must test negative initially but positive at enrollment, not be on oxygen therapy, and can't have had COVID-19 or a vaccine in the last 90 days unless immunocompromised.

Inclusion Criteria

Asymptomatic contact of an individual with laboratory confirmed SARS-CoV-2 infection
I have two or more symptoms that are moderate to severe.
I tested negative for COVID-19 recently.
See 7 more

Exclusion Criteria

Pregnancy
Breastfeeding
I am using supplemental oxygen.
See 13 more

Timeline for a Trial Participant

Screening

Participants are screened for eligibility to participate in the trial

2-4 weeks

Early Treatment

Participants receive Upamostat 400 mg or placebo orally once daily for 14 days

2 weeks
Daily follow-up via symptom questionnaire

Post-Exposure Prophylaxis

Participants are monitored for incidence of symptomatic COVID-19

2 weeks
Daily follow-up via symptom questionnaire

Follow-up

Participants are monitored for safety and effectiveness after treatment

12 weeks
Weekly follow-up via symptom questionnaire

What Are the Treatments Tested in This Trial?

Interventions

  • Placebo
  • Upamostat
Trial Overview The PROTECT-APT 1 study tests Upamostat against a placebo as an early treatment and preventative measure for COVID-19. Participants are randomly assigned to receive either the drug or placebo without knowing which one they get, to compare safety and effectiveness.
How Is the Trial Designed?
2Treatment groups
Experimental Treatment
Placebo Group
Group I: Early Treatment: Upamostat 400 mgExperimental Treatment1 Intervention
Group II: Early Treatment: Placebo Oral CapsulePlacebo Group1 Intervention

Find a Clinic Near You

Who Is Running the Clinical Trial?

Henry M. Jackson Foundation for the Advancement of Military Medicine

Lead Sponsor

Trials
103
Recruited
94,300+

Joint Program Executive Office Chemical, Biological, Radiological, and Nuclear Defense Enabling Biotechnologies

Collaborator

Trials
3
Recruited
1,000+

RedHill Biopharma Limited

Industry Sponsor

Trials
20
Recruited
2,700+

FHI Clinical, Inc.

Collaborator

Trials
2
Recruited
380+

Citations

RedHill Announces Publication of Positive Phase 2 Study ...Positive data from a U.S. Phase 2 study of once-daily oral RHB-107 (upamostat) in symptomatic COVID-19 published in the peer-reviewed ...
RedHill Biopharma Secures Allowance of Key Chinese ...Further post-hoc analysis showed faster recovery periods from severe COVID-19 symptoms with a median of 3 days to recovery with RHB-107 compared ...
Phase 2/3 Study of Upamostat, a Serine Protease Inhibitor, ...One medication, remdesivir, has shown efficacy in treatment of COVID-19 in hospitalized patients with severe illness; several monoclonal ...
RedHill Announces Positive Phase 2 Study Results with ...Although not powered for efficacy assessment, the study showed highly promising efficacy results delivering a 100% reduction in hospitalization ...
5.pubmed.ncbi.nlm.nih.govpubmed.ncbi.nlm.nih.gov/37970658/
Upamostat: a serine protease inhibitor for antiviral, ...It has demonstrated preliminary evidence of efficacy against COVID-19, and nonclinical data suggest potential applicability against other viral illnesses, ...
Our Programs - Pipeline - RHB-107RHB-107 successfully completed a Phase 2 study in non-hospitalized symptomatic COVID-19 patients which evaluated the safety and tolerability profile of RHB ...
7.pubmed.ncbi.nlm.nih.govpubmed.ncbi.nlm.nih.gov/36549549/
A randomized, placebo-controlled pilot study of upamostat, ...Conclusion: Upamostat was well tolerated, shortened recovery time, and decreased new severe symptoms and hospitalization. Keywords: COVID-19; ...
Mesupron (upamostat) / Heidelberg Pharma, RedHill... COVID-19 Outpatient Study with RHB-107 (PRNewswire) - "RedHill Biopharma Ltd....announced that the first patient was dosed in its U.S. Phase 2/3 study of ...
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