Zanzalintinib for Kidney Cancer with Bone Metastases

(ZAMBONI Trial)

UG
Overseen ByUCSF Genitourinary Oncology Clinical Trials Recruitment
Age: 18+
Sex: Any
Trial Phase: Phase 2
Sponsor: Kelly Fitzgerald, MD
Must be taking: Bone-strengthening agents
Stay on Your Current MedsYou can continue your current medications while participating
No Placebo GroupAll trial participants will receive the active study treatment (no placebo)
Prior Safety DataThis treatment has passed at least one previous human trial

What You Need to Know Before You Apply

What is the purpose of this trial?

This trial tests the effectiveness of zanzalintinib for treating kidney cancer that has spread to the bones. Researchers aim to determine if this drug, combined with a bone-strengthening agent, can benefit patients whose cancer has progressed after trying other treatments, including at least one type of immune therapy. Suitable candidates have advanced kidney cancer with at least three bone metastases and have previously tried 1-3 other therapies. As a Phase 2 trial, this research measures how well the treatment works in an initial, smaller group, offering a chance to contribute to important advancements in cancer care.

Do I need to stop my current medications to join the trial?

The trial does not specify if you need to stop your current medications, but it does mention that certain medications, like small molecule kinase inhibitors and some anticoagulants, should be stopped before starting the study treatment. It's best to discuss your specific medications with the trial team.

Is there any evidence suggesting that zanzalintinib is likely to be safe for humans?

Research has shown that zanzalintinib is promising in terms of safety for patients with advanced kidney cancer. Patients have tolerated zanzalintinib well in studies, whether used alone or with other treatments like nivolumab. Specifically, the STELLAR-002 study found that the combination had manageable safety for those with untreated stage 4 kidney cancer, meaning side effects were not severe enough to outweigh the treatment's benefits.

Additionally, when used alone, zanzalintinib has shown promising results in shrinking tumors in patients who have already tried other treatments for clear cell kidney cancer. While specific side effects weren't detailed, "manageable safety" suggests that any side effects are generally not life-threatening or too difficult to handle.

This trial is in the second phase, indicating that zanzalintinib has already been tested for safety in humans. This offers some reassurance about its safety, but ongoing trials are still needed to confirm these findings.12345

Why do researchers think this study treatment might be promising?

Zanzalintinib is unique because it specifically targets kidney cancer with bone metastases, offering a novel approach compared to traditional treatments like tyrosine kinase inhibitors or immune checkpoint inhibitors. Unlike these standard options, Zanzalintinib is administered orally, providing a more convenient mode of delivery. Researchers are particularly excited about its potential to work alongside bone-strengthening agents, addressing both the cancer and its impact on the bones simultaneously. This dual approach could enhance patient quality of life by managing symptoms effectively while targeting the cancer itself.

What evidence suggests that zanzalintinib might be an effective treatment for kidney cancer with bone metastases?

Studies have shown that zanzalintinib, the investigational drug tested in this trial for kidney cancer with bone metastases, has promising results. In one study, 38% of patients experienced a reduction in cancer size, and 88% saw their cancer either shrink or stop growing. Although this trial focuses on zanzalintinib alone, previous research indicates that combining zanzalintinib with nivolumab increased the number of patients who saw their cancer shrink to 63%, with 90% experiencing either shrinkage or stability. These findings suggest that zanzalintinib effectively manages advanced kidney cancer, even when other treatments have failed.16789

Who Is on the Research Team?

KF

Kelly Fitzgerald, MD

Principal Investigator

University of California, San Francisco

Are You a Good Fit for This Trial?

This trial is for patients with advanced kidney cancer that has spread to the bones. They must have tried 1-3 previous treatments, including at least one immune-based therapy. It's not suitable for those who haven't had prior treatment or don't meet specific health requirements.

Inclusion Criteria

I have at least three bone metastases, and not all will be treated with radiation.
I am 18 years old or older.
My hepatitis B virus load is undetectable with treatment.
See 12 more

Exclusion Criteria

I haven't taken any non-prescription drugs for my condition in the last 2 weeks.
Participation in an experimental drug study within 28 days of study enrollment
History of severe allergic, anaphylactic, or other hypersensitivity reactions to chimeric or humanized antibodies or fusion proteins
See 17 more

Timeline for a Trial Participant

Screening

Participants are screened for eligibility to participate in the trial

2-4 weeks

Treatment

Participants receive 100 mg Zanzalintinib orally once a day in 28-day cycles, along with an investigator-choice bone-strengthening agent. Radiation therapy for symptomatic metastases is allowed.

Up to 24 months

Follow-up

Participants are monitored for safety, effectiveness, and survival after treatment, with assessments for progression-free survival and overall survival.

Up to 24 months

What Are the Treatments Tested in This Trial?

Interventions

  • Zanzalintinib
Trial Overview The study tests zanzalintinib combined with a bone-strengthening agent chosen by the investigator in people with metastatic renal cell carcinoma and bone involvement. Participants will also undergo CT scans, bone scans, and may receive non-experimental radiation therapy.
How Is the Trial Designed?
1Treatment groups
Experimental Treatment
Group I: Treatment (Zanzalintinib)Experimental Treatment5 Interventions

Find a Clinic Near You

Who Is Running the Clinical Trial?

Kelly Fitzgerald, MD

Lead Sponsor

Exelixis

Industry Sponsor

Trials
126
Recruited
20,500+
Michael M. Morrissey profile image

Michael M. Morrissey

Exelixis

Chief Executive Officer since 2010

PhD in Chemistry from Harvard University, BSc in Chemistry from the University of Wisconsin

Vicki L. Goodman profile image

Vicki L. Goodman

Exelixis

Chief Medical Officer since 2022

MD

Citations

Novel TKI Zanzalintinib Confers Promising Antitumor ...Patients with advanced clear cell renal cell carcinoma treated with zanzalintinib had experienced promising antitumor activity with manageable toxicity.
Study Details | NCT07043608 | Zanzalintinib for Metastatic ...This is a single-institution, phase 2 trial of zanzalintinib plus investigator-choice bone-strengthening agent in patients with metastatic renal cell carcinoma ...
Press Release - Exelixis, Inc.Results for Exelixis' next-generation tyrosine kinase inhibitor demonstrated an objective response rate of 38% and a disease control rate of 88% –.
STELLAR-304: a phase III study of zanzalintinib (XL092) plus ...Cabozantinib showed significant benefits in PFS (9.0 vs 5.6 months, respectively; HR for cabozantinib vs sunitinib: 0.60, 95% CI: 0.37–0.97; p = 0.019) and ...
Exelixis Announces Encouraging Results from Phase 1b/2 ...Zanzalintinib in combination with nivolumab demonstrated an objective response rate of 63% and a disease control rate of 90% ...
Press Release - Exelixis, Inc.Zanzalintinib in combination with nivolumab demonstrated an objective response rate of 63% and a disease control rate of 90%.
Biomarker analysis of zanzalintinib in clear cell renal ...Zanza in pts with advanced ccRCC leads to modulation of plasma biomarkers associated with angiogenesis and peripheral immune cell subsets.
Zanzalintinib/Nivolumab Combo Shows Promise in ...The STELLAR-002 study reports promising efficacy and manageable safety for zanzalintinib plus nivolumab in untreated stage 4 RCC patients.
Zanzalintinib a potential 'novel breakthrough' in advanced ...Zanzalintinib monotherapy showed promising antitumor activity among patients with previously treated clear cell renal cell carcinoma.
Unbiased ResultsWe believe in providing patients with all the options.
Your Data Stays Your DataWe only share your information with the clinical trials you're trying to access.
Verified Trials OnlyAll of our trials are run by licensed doctors, researchers, and healthcare companies.
Terms of Service·Privacy Policy·Cookies·Security