AZD4144 Safety Study in Healthy Subjects

No longer recruiting at 1 trial location
AC
Overseen ByAstraZeneca Clinical Study Information Center

What You Need to Know Before You Apply

What is the purpose of this trial?

This trial aims to understand the safety and effects of a new treatment called AZD4144. Researchers assess how the body processes AZD4144 and whether it causes any side effects, comparing it to a placebo (a harmless pill resembling the real treatment). They also examine how AZD4144 interacts with other drugs like rosuvastatin and furosemide. The trial suits healthy individuals, particularly those of Japanese or Chinese descent, who have not lived outside their country for more than ten years. Individuals with significant health issues or allergies may not be suitable for this trial. As a Phase 1 trial, the research focuses on understanding how the treatment works in people, offering participants the opportunity to be among the first to receive this new treatment.

Do I need to stop my current medications for the trial?

Yes, you will need to stop taking any prescribed or nonprescribed medications, as the trial excludes participants using these drugs.

Is there any evidence suggesting that AZD4144 is likely to be safe for humans?

Research shows that AZD4144 has undergone testing for safety and tolerability. Previous patients demonstrated that daily intake of AZD4144 is generally well-tolerated, with most side effects being mild and not serious.

The treatment targets a specific protein called NLRP3, and studies indicate it does so effectively without impacting other parts of the body. This suggests that AZD4144 might have fewer unwanted effects.

This study is in the early stages, focusing primarily on understanding safety in healthy individuals. Further studies will offer more information about its safety in larger groups.12345

Why are researchers excited about this trial's treatment?

Researchers are excited about AZD4144 because it offers a new approach to treatment by potentially enhancing the effects of medications like rosuvastatin and furosemide. Unlike existing treatments that focus on singular pathways, AZD4144 is being investigated for its ability to work synergistically with other drugs, possibly improving outcomes for patients. This novel mechanism of action could lead to more effective and comprehensive treatment strategies, setting it apart from current options.

What evidence suggests that AZD4144 could be effective?

Research has shown that AZD4144 blocks a protein called NLRP3, which causes inflammation. This protein is linked to conditions where inflammation plays a key role. Studies have found that AZD4144 effectively inhibits NLRP3, suggesting it might help with inflammation-related issues. In this trial, participants will receive either AZD4144 or a placebo to assess its safety and tolerability. Testing so far has shown that AZD4144 is safe and well-tolerated, with no major side effects in healthy individuals. Although information on its effectiveness for specific conditions in humans is limited, its mechanism offers promising potential for treating inflammation-driven diseases.12356

Are You a Good Fit for This Trial?

This trial is for healthy individuals who can participate in a three-part study. Specific eligibility criteria are not provided, but typically participants must meet certain health standards and not have conditions that could interfere with the study or pose risks.

Inclusion Criteria

For healthy Japanese cohorts: healthy male and female participants are to be Japanese, defined as having both parents and 4 grandparents who are Japanese. This includes second and third generation participants of Japanese descent whose parents or grandparents are living in a country other than Japan
I am a man who can father children and will use birth control.
I am a woman who cannot become pregnant, confirmed at my screening visit.
See 4 more

Exclusion Criteria

I have a condition that makes me more likely to get infections.
Any positive result on Screening for serum Hepatitis B surface antigen (HBsAg), anti-Hepatitis B core (HBc), hepatitis C antibody, or Human immunodeficiency virus (HIV)
Any clinically important abnormalities in ECG
See 10 more

Timeline for a Trial Participant

Screening

Participants are screened for eligibility to participate in the trial

4 weeks

Treatment Part A

Participants receive a single ascending dose of AZD4144 or placebo

4 days
Residential stay from Day -1 to Day 4

Treatment Part B

Participants receive multiple ascending doses of AZD4144 or placebo

15 days
Residential stay from Day -1 to Day 15

Treatment Part C

Participants receive rosuvastatin and furosemide with and without AZD4144 to assess drug-drug interactions

12 days
Residential stay from Day -1 to Day 3 and Day 9 to Day 12

Follow-up

Participants are monitored for safety and effectiveness after treatment

3 days after last dose
Final follow-up visit on Day 10+3 for Part A and Day 20+3 for Part B and C

What Are the Treatments Tested in This Trial?

Interventions

  • AZD4144
Trial Overview The trial tests AZD4144's safety, tolerability, how it's processed by the body (pharmacokinetics), and its effects on the body (pharmacodynamics) compared to a placebo. It also examines if AZD4144 affects how rosuvastatin, a cholesterol medication, works when both drugs are taken together.
How Is the Trial Designed?
17Treatment groups
Experimental Treatment
Placebo Group
Group I: Part C cohort- Treatment C2Experimental Treatment1 Intervention
Group II: Part C Cohort- Treatment C1Experimental Treatment1 Intervention
Group III: Part B2- Japanese CohortExperimental Treatment1 Intervention
Group IV: Part B1- Cohort 3Experimental Treatment1 Intervention
Group V: Part B1- Cohort 2Experimental Treatment1 Intervention
Group VI: Part B1- Cohort 1Experimental Treatment1 Intervention
Group VII: Part A3-Chinese CohortExperimental Treatment1 Intervention
Group VIII: Part A2: Japanese Cohort 2Experimental Treatment1 Intervention
Group IX: Part A2-Japanese cohort 1Experimental Treatment1 Intervention
Group X: Part A1-Cohort 3Experimental Treatment1 Intervention
Group XI: Part A1-Cohort 1Experimental Treatment1 Intervention
Group XII: Part A1- Cohort 2Experimental Treatment1 Intervention
Group XIII: Part A3- PlaceboPlacebo Group1 Intervention
Group XIV: Part B2- PlaceboPlacebo Group1 Intervention
Group XV: Part A1- PlaceboPlacebo Group1 Intervention
Group XVI: Part B1- PlaceboPlacebo Group1 Intervention
Group XVII: Part A2- PlaceboPlacebo Group1 Intervention

Find a Clinic Near You

Who Is Running the Clinical Trial?

AstraZeneca

Lead Sponsor

Trials
4,491
Recruited
290,540,000+

Sir Pascal Soriot

AstraZeneca

Chief Executive Officer since 2012

Veterinary Medicine from École nationale vétérinaire d'Alfort, MBA from HEC Paris

Dr. Cristian Massacesi

AstraZeneca

Chief Medical Officer since 2021

MD from Marche Polytechnic University, Oncology training at Royal Marsden Hospital, Kaplan Comprehensive Cancer Center, and European Institute of Oncology

Pascal Soriot

AstraZeneca

Chief Executive Officer since 2012

Veterinary Medicine from École nationale vétérinaire d'Alfort, MBA from HEC Paris

Cristian Massacesi

AstraZeneca

Chief Medical Officer since 2021

MD from Marche Polytechnic University, Medical Oncology training at Royal Marsden Hospital, Kaplan Comprehensive Cancer Center, and European Institute of Oncology

Citations

NCT06491550 | A Study to Assess the Safety, Tolerability ...This study will compare the safety, tolerability, pharmacokinetics (PK), and pharmacodynamics (PD) of AZD4144 with placebo in healthy participants.
A study to investigate the safety, tolerability and ...The aim of this study is to evaluate the safety and tolerability, and pharmacodynamics (PD) of AZD4144 administered as repeated daily oral dosing.
Discovery of AZD4144, a Selective and Potent NLRP3 ...The compound inhibits NLRP3 selectively with high potency, has beneficial pharmacokinetic properties, and shows a favorable off-target pharmacology profile.
NCT07215702 | A Study to Investigate the Efficacy, Safety, ...The main goal is to compare specific kidney function measurements between those participants receiving AZD4144 and those receiving the placebo.
AZD4144 Safety Study in Healthy SubjectsThis study consists of 3 parts: Part A, Part B and Part C. This study will compare the safety, tolerability, pharmacokinetics (PK), and pharmacodynamics ...
NCT06925854 | A Study to Investigate How AZD4144 ...A Study to Investigate How AZD4144 Affects the Pharmacokinetics of Rosuvastatin in Healthy Participants. ClinicalTrials.gov ID NCT06925854.
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