222 Participants Needed

177Lu-FAP-2286 for Solid Cancers

(LuMIERE Trial)

Recruiting at 23 trial locations
CO
NP
Overseen ByNovartis Pharmaceuticals
No Placebo GroupAll trial participants will receive the active study treatment (no placebo)

What You Need to Know Before You Apply

What is the purpose of this trial?

This trial explores a new treatment called 177Lu-FAP-2286, a radiopharmaceutical therapy, for individuals with certain types of solid tumors. The goal is to assess the safety and efficacy of this treatment, particularly for pancreatic, lung, and breast cancers. The first part of the trial tests different doses to identify the safest one, while the second part evaluates its effectiveness both alone and with chemotherapy. Participants should have a solid tumor resistant to other treatments and must have tumors expressing a specific protein called FAP, verified through imaging. This trial may suit those whose cancer has not responded to standard therapies and who have specific types of pancreatic, lung, or breast cancer. As a Phase 1, Phase 2 trial, this study aims to understand how the treatment works in people and measure its effectiveness in an initial, smaller group.

Will I have to stop taking my current medications?

The trial protocol does not specify if you need to stop taking your current medications. However, you should discuss your current medications with the study team to ensure they don't interfere with the trial treatments.

Will I have to stop taking my current medications?

The trial does not specify if you need to stop taking your current medications. However, you should not have received certain anticancer treatments within 14 to 28 days before starting the trial, depending on the type of treatment. It's best to discuss your current medications with the trial team to ensure they don't interfere with the study.

Is there any evidence suggesting that 177Lu-FAP-2286 is likely to be safe for humans?

Research has shown that 177Lu-FAP-2286 has generally been well-tolerated in earlier studies. In these studies, participants with various advanced or metastatic solid tumors received the treatment, and early results indicated its safety. While some side effects occurred, they were mostly mild to moderate and manageable, such as tiredness or nausea, which are common with many cancer treatments.

This treatment remains in the early testing phase, which aims to ensure safety and determine the correct dosage for future studies. So far, the safety results appear promising, but ongoing studies will continue to monitor and gather more information about its safety.12345

Why are researchers excited about this study treatment?

Researchers are excited about 177Lu-FAP-2286 because it introduces a new way to target solid tumors. Unlike traditional therapies that often affect both healthy and cancerous cells, 177Lu-FAP-2286 specifically targets fibroblast activation protein (FAP), which is commonly found in cancerous tumors. This precision targeting could potentially minimize damage to healthy tissues and improve treatment outcomes. Additionally, the use of the radioactive isotope Lutetium-177 allows for both imaging and treatment, providing a dual benefit in managing cancer. These unique features make 177Lu-FAP-2286 a promising option for patients with solid tumors.

What evidence suggests that 177Lu-FAP-2286 might be an effective treatment for solid cancers?

Research has shown that 177Lu-FAP-2286 holds promise for treating solid cancers. It targets fibroblast activation protein (FAP), commonly found in tumors but not in normal tissues, allowing it to attack cancer cells while sparing healthy ones. Studies indicate it has a manageable safety profile, causing few serious side effects. In this trial, participants will join different phases: the Phase 1 Dose Escalation arm will include up to 30 patients with solid tumors, while the Phase 2 arm will treat up to 192 participants with 177Lu-FAP-2286 in tumor-specific groups, both as monotherapy and in combination with chemotherapy. Early results from patients with advanced tumors suggest it could be a hopeful treatment option.12567

Who Is on the Research Team?

NP

Novartis Pharmaceuticals

Principal Investigator

Novartis Pharmaceuticals

Are You a Good Fit for This Trial?

This trial is for adults with advanced solid tumors that have worsened after treatment or don't respond to it. They should be in good physical condition, not pregnant, and willing to use contraception. People with active secondary cancers, brain metastases, recent cancer treatments or surgeries, ongoing serious side effects from past treatments (except hair loss), severe urinary issues, known allergies to scan contrast media, infections needing antibiotics recently, significant heart problems are excluded.

Inclusion Criteria

Have a life expectancy of ≥ 6 months
My cancer has returned or spread and this is confirmed by tests.
Have measurable disease per RECIST v1.1 meeting specific criteria
See 5 more

Exclusion Criteria

Inability to complete needed investigational and standard imaging examinations
I have heart problems that affect my daily activities.
I have lost a lot of weight recently.
See 12 more

Timeline for a Trial Participant

Screening

Participants are screened for eligibility to participate in the trial

2-4 weeks
1 visit (in-person)

Treatment

Participants receive a single IV dose of [177Lu]Lu FAP 2286 every 6 weeks in Phase 1 and every 4 weeks in Phase 2, up to a maximum of 6 doses

24-36 weeks
Visits every 4-6 weeks for treatment and assessments

End of Treatment (EOT) Visit

Participants have an EOT visit 6-8 weeks after the last dose in Phase 1 and within 28 days in Phase 2

6-8 weeks
1 visit (in-person)

Post Treatment Safety Follow-up

Participants undergo safety follow-up for 6 weeks after discontinuation of study treatment

6 weeks
1 visit (in-person or virtual)

Long-term Follow-up (LTFU) Period

Participants are monitored for safety, disease, and survival assessments every 12 weeks for 2 years, then every 6 months until 5 years

5 years
Visits every 12 weeks for 2 years, then every 6 months

What Are the Treatments Tested in This Trial?

Interventions

  • 177Lu-FAP-2286
Trial Overview The study tests the safety and ideal dose of a new drug called 177Lu-FAP-2286 in Phase 1 and its effectiveness at shrinking tumors in Phase 2. Patients must have specific FAP-expressing tumor types for Phase 2. The response rate will be measured using standard criteria.
How Is the Trial Designed?
2Treatment groups
Experimental Treatment
Group I: Phase 2: Specific Solid TumorsExperimental Treatment2 Interventions
Group II: Phase 1: Dose EscalationExperimental Treatment2 Interventions

Find a Clinic Near You

Who Is Running the Clinical Trial?

Clovis Oncology, Inc.

Lead Sponsor

Trials
65
Recruited
11,100+

Patrick J. Mahaffy

Clovis Oncology, Inc.

Chief Executive Officer since 2009

BA from Haverford College, MBA from Columbia University

Lindsey Rolfe

Clovis Oncology, Inc.

Chief Medical Officer since 2015

Specialist accreditation in pharmaceutical medicine

Novartis Pharmaceuticals

Lead Sponsor

Trials
2,963
Recruited
4,275,000+
Founded
1996
Headquarters
Basel, Switzerland
Known For
Precision medicine
Top Products
Gleevec, Cosentyx, Entresto, Kisqali
Dr. Vas Narasimhan profile image

Dr. Vas Narasimhan

Novartis Pharmaceuticals

Chief Executive Officer since 2018

MD from Harvard Medical School

Dr. Shreeram Aradhye profile image

Dr. Shreeram Aradhye

Novartis Pharmaceuticals

Chief Medical Officer since 2021

MD

Published Research Related to This Trial

The newly developed albumin binder-conjugated FAPI radiotracers, TEFAPI-06 and TEFAPI-07, showed significantly improved tumor accumulation and retention compared to the original FAPI tracer, enhancing their potential for cancer treatment.
Both TEFAPI-06 and TEFAPI-07 demonstrated remarkable tumor growth inhibition in pancreatic cancer models with negligible side effects, indicating their promise for future clinical applications.
Albumin Binder-Conjugated Fibroblast Activation Protein Inhibitor Radiopharmaceuticals for Cancer Therapy.Xu, M., Zhang, P., Ding, J., et al.[2023]
The study evaluated two radiopharmaceuticals, [177Lu]Lu-DOTA.SA.FAPi and [177Lu]Lu-DOTAGA.(SA.FAPi)2, in patients with various cancers, showing that [177Lu]Lu-DOTAGA.(SA.FAPi)2 had significantly higher tumor absorbed doses and longer effective half-lives, indicating its potential for better therapeutic efficacy.
Both agents demonstrated safety in administration, with biodistribution observed in various organs, but [177Lu]Lu-DOTAGA.(SA.FAPi)2 showed superior pharmacokinetics, making it a promising candidate for treating end-stage cancer patients using a theranostic approach.
First-In-Human Results on the Biodistribution, Pharmacokinetics, and Dosimetry of [177Lu]Lu-DOTA.SA.FAPi and [177Lu]Lu-DOTAGA.(SA.FAPi)2.Ballal, S., Yadav, MP., Moon, ES., et al.[2021]
The novel radiopharmaceutical agent 177Lu-DOTA-DG was successfully synthesized with a high radiochemical yield and demonstrated excellent stability in human serum for up to 120 hours, indicating its potential for safe use in cancer imaging and therapy.
In preclinical studies, 177Lu-DOTA-DG caused significantly more DNA damage in cancer cells compared to untreated cells, suggesting its efficacy as a targeted treatment for cancer tissues.
In vivo and in vitro evaluation of 177Lu-labeled DOTA-2-deoxy-D-glucose in mice. A novel radiopharmaceutical agent for cells imaging and therapy.Zhang, J., Wang, Z., Liu, H., et al.[2019]

Citations

NCT04939610 | A Study of 177Lu-FAP-2286 in Advanced ...Phase 1 of this study is designed to evaluate the safety and establish the recommended intravenous (IV) Phase 2 dose (RP2D) for [177Lu]Lu FAP 2286 monotherapy ...
177Lu-FAP-2286 in patients with advanced or metastatic solid ...177Lu-FAP-2286 in patients with advanced or metastatic solid tumors: Initial data from a phase 1/2 study investigating safety, pharmacokinetics, ...
Current clinical application of lutetium‑177 in solid tumors ...As a result, 177Lu can be used for both diagnosis and treatment for diseases such as prostatic and gastric cancer. Therefore, based on the available data, the ...
177Lu-FAP-2286 Displays Preliminary Antitumor Activity in ...Lutetium-177-FAP-2286 produced preliminary evidence of antitumor activity with a manageable safety profile in patients with advanced or metastatic solid tumors.
[177Lu]Lu-FAPI Radioligand Therapy: Emerging Horizons ...[177Lu]Lu-FAPI Radioligand Therapy: Emerging Horizons and Clinical Promise in Solid Tumors: A Comprehensive Review · Background: Overview of FAPI.
A Study of 177Lu-FAP-2286 in Advanced Solid Tumors ...Phase 2 is designed to evaluate the safety and efficacy of [177Lu]Lu FAP 2286 as monotherapy in participants with pancreatic ductal ...
LuMIERE: A Phase 1/2, Multicenter, Open-label, Non ...The purpose of this study is to test the safety of the experimental drugs called 68Ga-FAP-2286 and 177Lu-FAP-2286.
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