73 Participants Needed

NTX-253 for Schizophrenia

DF
LC
Overseen ByLisa Corey
Age: 18 - 65
Sex: Any
Trial Phase: Phase < 1
Sponsor: Neurosterix
Must be taking: Antipsychotics
No Placebo GroupAll trial participants will receive the active study treatment (no placebo)

What You Need to Know Before You Apply

What is the purpose of this trial?

This trial aims to test a new treatment called NTX-253, a potential drug for schizophrenia, to assess its safety, tolerability, and how the body processes it. The study includes different groups: some will receive NTX-253, while others will receive a placebo (a pill with no active drug) in varying doses. It seeks adults with stable schizophrenia whose symptoms are under control and who are not resistant to treatment. Those with stable schizophrenia may find this trial suitable. As a Phase 1 trial, participants will be among the first to receive this new treatment, helping researchers understand its effects in people.

Will I have to stop taking my current medications?

The trial information does not specify if you need to stop taking your current medications. It's best to discuss this with the trial coordinators or your doctor.

Is there any evidence suggesting that NTX-253 is likely to be safe for humans?

Research has shown that NTX-253 looks promising in early studies. Initial tests found it safe, as animals tolerated it well without major side effects. However, NTX-253 is just beginning its first human trials. This phase primarily assesses safety and tolerability in people. While the results are promising, human trials are necessary to confirm safety. Researchers will closely monitor for any side effects to determine how safe NTX-253 is for humans.12345

Why do researchers think this study treatment might be promising for schizophrenia?

Researchers are excited about NTX-253 for schizophrenia because it offers a novel approach compared to current treatments like antipsychotics, which primarily target dopamine receptors. NTX-253 potentially works through a different mechanism, which might provide benefits for patients who do not respond well to existing therapies. This new treatment could lead to better management of symptoms with fewer side effects, making it a promising option for those with schizophrenia.

What evidence suggests that NTX-253 might be an effective treatment for schizophrenia?

Research has shown that NTX-253 is a promising new treatment for schizophrenia. It targets a specific part of the brain to control symptoms like hallucinations and delusions. This method differs from traditional medications and might be safer and more effective. Early studies suggest that NTX-253 can help balance brain signals, potentially reducing these symptoms. Although more research is needed, NTX-253 could improve outcomes for people with schizophrenia, making it an exciting option. Participants in this trial will receive NTX-253 in various dosing regimens to further evaluate its effectiveness and safety.12456

Who Is on the Research Team?

DF

Doug Feltner, MD

Principal Investigator

Neurosterix

Are You a Good Fit for This Trial?

This trial is for adults aged 18-55, both healthy and those with stable schizophrenia. Participants must not be pregnant or breastfeeding, should either live a truly abstinent lifestyle or use birth control, and have a BMI within specified ranges (17.5 to 36.0 kg/m2). Those with schizophrenia must have a PANSS score less than 80.

Inclusion Criteria

I am a male or a female not able to have children, aged 18-55, and either not sexually active or using birth control.
My BMI is between 18.0 and 30.0.
My schizophrenia is stable.
See 4 more

Timeline for a Trial Participant

Screening

Participants are screened for eligibility to participate in the trial

2-4 weeks

Single Ascending Dose (SAD)

Participants receive a single ascending dose of NTX-253 or placebo, including a food effect cohort and a CSF cohort in healthy volunteers

8 days
Multiple visits for dosing and monitoring

Multiple Ascending Dose (MAD)

Participants receive multiple ascending doses of NTX-253 or placebo for 10 consecutive days, including cohorts with stable schizophrenic participants

10 days
Daily visits for dosing

Follow-up

Participants are monitored for safety and effectiveness after treatment

4 weeks
Follow-up visits at Day 17 for healthy volunteers and Day 35 for participants with stable schizophrenia

What Are the Treatments Tested in This Trial?

Interventions

  • NTX-253

Trial Overview

The study tests the safety and how the body processes NTX-253 when taken orally by healthy adults and adults with stable schizophrenia. It compares NTX-253 against a placebo in different groups of participants over single and multiple doses.

How Is the Trial Designed?

5

Treatment groups

Experimental Treatment

Group I: Placebo Part 2Experimental Treatment1 Intervention
Group II: Placebo Part 1aExperimental Treatment1 Intervention
Group III: NTX-253 Part 2Experimental Treatment1 Intervention
Group IV: NTX-253 Part 1bExperimental Treatment1 Intervention
Group V: NTX-253 Part 1aExperimental Treatment1 Intervention

Find a Clinic Near You

Who Is Running the Clinical Trial?

Neurosterix

Lead Sponsor

Citations

Single and Multiple Ascending Doses of NTX-253 in ...

This study will assess the safety, tolerability, and pharmacokinetics of NTX-253 following oral administration in both healthy adult ...

Addex Spin-Out Neurosterix has started a Phase 1 Clinical ...

NTX-253 is a potent, selective, orally available PAM of M4 that fine-tunes muscarinic signaling with the potential to reduce psychosis symptoms ...

Neurosterix Announces Phase 1 Study of NTX-253 for ...

NTX-253 enters phase 1 trials, exploring a novel approach to schizophrenia treatment with potential for improved safety and efficacy.

Addex Spin-Out Neurosterix Begins Phase 1 Trial of Novel ...

NTX-253 is a potent, selective, orally available positive allosteric modulator (PAM) of the muscarinic M4 receptor. Unlike traditional ...

NTX-253 for Schizophrenia

The study tests the safety and how the body processes NTX-253 when taken orally by healthy adults and adults with stable schizophrenia. It compares NTX-253 ...

Addex Spin-Out Neurosterix has started a Phase 1 Clinical ...

NTX-253 is a potent, selective, orally available PAM of M4 that fine-tunes muscarinic signaling with the potential to reduce psychosis symptoms ...